SCHEMBL5544973

SCHEMBL5544973

CCc1ccc(C(=O)NC2N=CC3=CN(S(=O)(=O)c4ccsc4)CCC3=N2)cc1

nearest known ligand 0.33

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.32
OPRM1 P35372 1/20 0.31
OPRD1 P41143 1/20 0.31
OPRK1 P41145 1/20 0.31
ALDH1A1 P00352 3/20 0.31
DRD2 P14416 3/20 0.31
DRD4 P21917 3/20 0.31
MEN1 O00255 1/20 0.31
POLB P06746 1/20 0.31
KMT2A Q03164 1/20 0.31
PLK1 P53350 1/20 0.31
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5545055 0.85 ALDH1A1 (0.43) GAAALDH1A1MEN1POLBKMT2A
SCHEMBL5545093 0.82 HSD11B1 (0.35) OPRM1OPRD1OPRK1MEN1POLB
SCHEMBL5538108 0.79 PKM (0.42) OPRK1ALDH1A1
SCHEMBL5548484 0.76 KMT2A (0.54) GAAALDH1A1MEN1POLBKMT2A
SCHEMBL5540250 0.75 LMNA (0.39) OPRK1DRD2DRD4MEN1POLB
SCHEMBL5546899 0.74 ALDH1A1 (0.48) GAAALDH1A1MEN1POLBKMT2A
SCHEMBL5540347 0.72 CCKAR (0.39) ALDH1A1MEN1KMT2A
SCHEMBL5546891 0.71 KMT2A (0.39) GAAALDH1A1POLBKMT2A
SCHEMBL5546586 0.70 HTR3A (0.41) PLK1
SCHEMBL5546858 0.67 MEN1 (0.38) ALDH1A1MEN1KMT2APLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007534719-A 2007-11-29 JP claimed
EP-1742925-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2007-01-17 EP claimed
WO-2005105759-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2005-11-10 WO claimed