Acridine

Acridine

SCHEMBL557520

NCCCCCC(=O)O.c1ccc2nc3ccccc3cc2c1

nearest known ligand 0.53

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

PLATPLG

The experimentally established mechanism targets of Acridine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLG known ✓ P00747 1/20 0.53
ALDH1A1 P00352 3/20 0.53
KMT2A Q03164 3/20 0.53
MEN1 O00255 2/20 0.53
LMNA P02545 2/20 0.53
THRB P10828 2/20 0.53
ALOX15 P16050 2/20 0.53
SLC6A2 P23975 1/20 0.53
RECQL P46063 1/20 0.53
SLC6A3 Q01959 1/20 0.53
CYP2D6 P10635 1/20 0.50
NFKB1 P19838 1/20 0.50
NPSR1 Q6W5P4 3/20 0.48
BLM P54132 2/20 0.48
MAPT P10636 2/20 0.47
GLA P06280 1/20 0.47
HPGD P15428 1/20 0.47
ACHE P22303 1/20 0.47
LTB4R Q15722 3/20 0.45
HDAC3 O15379 3/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Naphthalene SCHEMBL6898872 0.85 LMNA (0.68) ALDH1A1KMT2AMEN1LMNATHRB
Acridine SCHEMBL17892439 0.84 PPARG (0.53) ALDH1A1KMT2AMEN1ALOX15MAPT
Acridine SCHEMBL28897857 0.83 ALDH1A1 (0.62) ALDH1A1KMT2AMEN1LMNANPSR1
Acridine SCHEMBL27894463 0.83 MAPT (0.68) ALDH1A1KMT2AMEN1LMNAMAPT
Acridine SCHEMBL9542382 0.81 AKR1B1 (0.50) ALDH1A1KMT2AMEN1ALOX15MAPT
Acridine SCHEMBL9614417 0.76 ALDH1A1 (0.58) ALDH1A1KMT2AMEN1LMNACYP2D6
Acridine SCHEMBL4854060 0.75 ALDH1A1 (0.68) ALDH1A1KMT2AMEN1LMNAMAPT
5-Aminovaleric Acid SCHEMBL11669034 0.75 NFKB1 (0.89) ALDH1A1KMT2AMEN1LMNATHRB
Behenic Acid SCHEMBL31536707 0.73 GPR84 (0.61) ALDH1A1KMT2AMEN1LMNAALOX15
Benzamide SCHEMBL14574628 0.73 LMNA (0.61) ALDH1A1KMT2AMEN1LMNATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120035320-A1 POLYACRIDINE NUCLEIC ACID DELIVERY PEPTIDE COMPLEXES UNIVERSITY OF IOWA RESEARCH FOUNDATION (US) 2012-02-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120035320-A1 POLYACRIDINE NUCLEIC ACID DELIVERY PEPTIDE COMPLEXES NUP205, PABPC1, SARNP PLG 1586/4885ALDH1A1 3315/4885KMT2A 2891/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.