SCHEMBL557722

SCHEMBL557722

CCOC(OCC)C(=N)OC

nearest known ligand 0.38

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.38
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21011290 0.89 THRB (0.31) THRB
SCHEMBL17615951 0.79
SCHEMBL18056899 0.74 THRB (0.31) THRB
SCHEMBL559834 0.73
SCHEMBL11289833 0.71 THRB (0.42) THRBLMNA
SCHEMBL14867667 0.71 THRB (0.42) THRBLMNA
SCHEMBL18039126 0.70 THRB (0.36) THRBLMNA
SCHEMBL27367061 0.70 THRB (0.36) THRBLMNA
SCHEMBL13814227 0.70 THRB (0.36) THRBLMNA
SCHEMBL558811 0.69 THRB (0.40) THRBLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 296 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-7126254-A None JP disclosed
US-12637428-B2 Isoquinoline derivatives as SIK2 inhibitors CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2026-05-26 US disclosed
EP-4211119-B1 2-AMINOQUINAZOLINES AS LRRK2 INHIBITORS, PHARMACEUTICAL COMPOSITIONS, AND USES THEREOF MERCK SHARP & DOHME LLC (US) 2026-05-13 EP disclosed
US-20260115297-A1 HETEROBIFUNCTIONAL COMPOUNDS AS DEGRADERS OF HPK1 ICAHN SCHOOL MED MOUNT SINAI (US) 2026-04-30 US disclosed
EP-4720057-A2 COMPOUNDS AND COMPOSITIONS AS CBP/P300 DEGRADERS AND USES THEREOF Oncopia Therapeutics, Inc. D/B/A SK Life Science Labs (US) 2026-04-08 EP disclosed
US-12570640-B2 2-aminoquinazolines as LRRK2 inhibitors, pharmaceutical compositions, and uses thereof MERCK SHARP & DOHME LLC (US) 2026-03-10 US disclosed
EP-3826722-B1 ISOQUINOLINE COMPOUNDS AND USES THEREOF HOFFMANN LA ROCHE (CH) 2026-02-18 EP disclosed
US-12516039-B2 N-linked isoquinoline amides as LRRK2 inhibitors, pharmaceutical compositions, and uses thereof MERCK SHARP & DOHME LLC (US) 2026-01-06 US disclosed
US-12473301-B2 Isoquinoline compounds for the treatment of cancer GENENTECH, INC. (US) 2025-11-18 US disclosed
US-12465648-B2 Heterobifunctional compounds as degraders of HPK1 ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI (US) 2025-11-11 US disclosed
US-7151105-B2 Inhibitors of Hepatitis C virus RNA-dependent RNA polymerase, and compositions and treatments using the same AGOURON PHARMACEUTICALS, INC. (US) 2006-12-19 US disclosed
US-20060122399-A1 Inhibitors of hepatitis C virus RNA-dependent RNA polymerase, and compositions and treatments using the same AGOURON PHARMACEUTICALS, INC. 2006-06-08 US disclosed
WO-2006018725-A1 INHIBITORS OF HEPATITIS C VIRUS RNA-DEPENDENT RNA POLYMERASE, AND COMPOSITIONS AND TREATMENTS USING THE SAME PFIZER INC. (US) 2006-02-23 WO disclosed
US-20050090501-A1 Heteroaryl-cyclic acetals AVENTIS PHARMA LIMITED (GB) 2005-04-28 US disclosed
EP-1140916-B1 HETEROARYL-CYCLIC ACETALS AVENTIS PHARMA LTD (GB) 2002-11-13 EP disclosed
EP-1218355-A1 THERAPEUTIC QUINAZOLINE DERIVATIVES AstraZeneca AB (SE) 2002-07-03 EP disclosed
EP-1140916-A1 HETEROARYL-CYCLIC ACETALS Aventis Pharma Limited (GB) 2001-10-10 EP disclosed
WO-2001021597-A1 THERAPEUTIC QUINAZOLINE DERIVATIVES ASTRAZENECA AB (SE) 2001-03-29 WO disclosed
WO-2000035911-A1 HETEROARYL-CYCLIC ACETALS AVENTIS PHARMA LIMITED (GB) 2000-06-22 WO disclosed
JP-H07126254-A IMIDAZOLE COMPOUND AND ITS PRODUCTION ISHIHARA SANGYO KAISHA LTD 1995-05-16 JP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12473301-B2 Isoquinoline compounds for the treatment of cancer PGK1, PHKG1, NEK1 THRB 4194/4885LMNA 3495/4885
US-12465648-B2 Heterobifunctional compounds as degraders of HPK1 HIPK1, MCL1, HYPK THRB 3105/4885LMNA 3665/4885
US-12637428-B2 Isoquinoline derivatives as SIK2 inhibitors SIK2, SIK1, SIK3 THRB 565/4885LMNA 1978/4885
US-12570640-B2 2-aminoquinazolines as LRRK2 inhibitors, pharmaceutical compositions, and uses thereof LRRK2, PARK7, CLK2 THRB 2517/4885LMNA 1809/4885
US-20060122399-A1 Inhibitors of hepatitis C virus RNA-dependent RNA polymerase, and compositions and treatments using the same RNASE1, GTF3C4, POLRMT THRB 4490/4885LMNA 2519/4885
US-20260115297-A1 HETEROBIFUNCTIONAL COMPOUNDS AS DEGRADERS OF HPK1 TTK, ITK, CLK1 THRB 2390/4885LMNA 3897/4885
US-20050090501-A1 Heteroaryl-cyclic acetals TNF, TNFRSF1A, CD40 THRB 1579/4885LMNA 919/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.