SCHEMBL5599096

SCHEMBL5599096

CCCC[C@H]1N(C(=O)c2ccccc2Cl)c2ccc(F)cc2C12CCNCC2

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GNRHR P30968 4/20 0.41
KCNH2 Q12809 1/20 0.41
RXFP1 Q9HBX9 1/20 0.38
SMYD3 Q9H7B4 2/20 0.35
HSD11B1 P28845 1/20 0.35
P2RX7 Q99572 4/20 0.34
PDK1 Q15118 3/20 0.33
PDK2 Q15119 3/20 0.33
PDK3 Q15120 3/20 0.33
PDK4 Q16654 3/20 0.33
MEN1 O00255 1/20 0.33
CRHBP P24387 1/20 0.33
KMT2A Q03164 1/20 0.33
CRHR2 Q13324 1/20 0.33
HPGD P15428 1/20 0.33
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5599389 0.86 GNRHR (0.40) GNRHRKCNH2RXFP1HSD11B1P2RX7
SCHEMBL5599374 0.86 GNRHR (0.40) GNRHRKCNH2RXFP1HSD11B1P2RX7
SCHEMBL5786887 0.85 GNRHR (0.41) GNRHRKCNH2RXFP1HSD11B1P2RX7
SCHEMBL5599203 0.85 GNRHR (0.39) GNRHRKCNH2RXFP1HSD11B1P2RX7
SCHEMBL5599816 0.81 TP53 (0.38) GNRHRKCNH2SMYD3MEN1KMT2A
SCHEMBL5599382 0.81 AGTR2 (0.36) GNRHRKCNH2MEN1KMT2A
SCHEMBL5782306 0.77 HTR2A (0.40) GNRHRKCNH2SMYD3HSD11B1
SCHEMBL5782925 0.76 LMNA (0.39) HSD11B1MEN1KMT2A
SCHEMBL5599289 0.75 DRD2 (0.37) GNRHRKCNH2SMYD3P2RX7HPGD
SCHEMBL5784243 0.75 GNRHR (0.42) GNRHRKCNH2SMYD3HSD11B1PDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005063745-A9 NOVEL SPIROINDOLINE OR SPIROISOQUINOLINE COMPOUNDS, METHODS OF USE AND COMPOSITIONS THEREOF ARENA PHARM INC (US) 2007-02-01 WO claimed