SCHEMBL5599231

SCHEMBL5599231

COc1ccc(C(=O)N2c3ccc(F)cc3C3(CCNCC3)[C@H]2Cc2ccc(OC)c(OC)c2)cc1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.42
KMT2A Q03164 5/20 0.41
MEN1 O00255 3/20 0.41
LMNA P02545 3/20 0.39
HTT P42858 3/20 0.39
NPC1 O15118 1/20 0.39
TP53 P04637 2/20 0.39
MCHR1 Q99705 1/20 0.38
KDM4E B2RXH2 1/20 0.37
POLB P06746 1/20 0.37
GFER P55789 1/20 0.36
ALDH1A1 P00352 3/20 0.36
THRB P10828 1/20 0.36
ALOX12 P18054 1/20 0.36
HCRTR1 O43613 1/20 0.36
HCRTR2 O43614 1/20 0.36
GLA P06280 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5820191 0.90 TDP2 (0.40) TSHRKMT2AMEN1LMNAHTT
SCHEMBL5788788 0.83 ALDH1A1 (0.38) TSHRKMT2AMEN1LMNAHTT
SCHEMBL5783676 0.76 ALDH1A1 (0.46) TSHRLMNAHTTMCHR1KDM4E
SCHEMBL5782925 0.72 LMNA (0.39) KMT2AMEN1LMNAHTTKDM4E
SCHEMBL5599203 0.72 GNRHR (0.39) NPC1ALDH1A1
SCHEMBL5780895 0.72 PSEN1 (0.40)
SCHEMBL4761766 0.70 PAX8 (0.37) TSHRLMNAALDH1A1MAPT
SCHEMBL5578809 0.69 KMT2A (0.55) TSHRKMT2AMEN1KDM4EPOLB
SCHEMBL5599578 0.69 HSD11B1 (0.40) HTTPOLBALDH1A1MAPT
SCHEMBL5784445 0.69 KDM4E (0.40) LMNAHTTTP53KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005063745-A9 NOVEL SPIROINDOLINE OR SPIROISOQUINOLINE COMPOUNDS, METHODS OF USE AND COMPOSITIONS THEREOF ARENA PHARM INC (US) 2007-02-01 WO claimed