SCHEMBL5600810

SCHEMBL5600810

O=C(c1ccc2c(c1)OCO2)[C@@H]1N(C(=O)c2ccc3c(c2)OCO3)c2ccccc2C12CCNCC2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.43
RAB9A P51151 2/20 0.43
ALDH1A1 P00352 6/20 0.42
TSHR P16473 6/20 0.42
LMNA P02545 2/20 0.42
USP2 O75604 1/20 0.42
HPGD P15428 8/20 0.41
HSD17B10 Q99714 2/20 0.41
GAA P10253 2/20 0.41
GFER P55789 1/20 0.41
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
TP53 P04637 1/20 0.40
KDM4E B2RXH2 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5599305 0.81 HPGD (0.41) NPC1RAB9AALDH1A1TSHRLMNA
SCHEMBL5782188 0.80 MEN1 (0.41) NPC1RAB9ALMNACYP3A4CYP2D6
SCHEMBL5599174 0.78 ALDH1A1 (0.46) ALDH1A1TSHRLMNAGAASMN1; SMN2
SCHEMBL5783881 0.72 TSHR (0.49) RAB9AALDH1A1TSHRHPGDGAA
SCHEMBL5599295 0.71 TSHR (0.47) ALDH1A1TSHRHPGDGAACYP3A4
SCHEMBL5786199 0.69 SIGMAR1 (0.43) ALDH1A1TSHRLMNACYP2C19SMN1; SMN2
SCHEMBL14638336 0.68 ALDH1A1 (0.56) NPC1RAB9AALDH1A1LMNAHPGD
SCHEMBL7464300 0.67 HPGD (0.75) NPC1ALDH1A1TSHRLMNAHPGD
SCHEMBL5599732 0.64 SMN1; SMN2 (0.38) ALDH1A1LMNAGAASMN1; SMN2NPSR1
SCHEMBL26413626 0.64 ALDH1A1 (0.47) NPC1RAB9AALDH1A1TSHRHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005063745-A9 NOVEL SPIROINDOLINE OR SPIROISOQUINOLINE COMPOUNDS, METHODS OF USE AND COMPOSITIONS THEREOF ARENA PHARM INC (US) 2007-02-01 WO claimed