SCHEMBL56219

SCHEMBL56219

CC(C)(C)OC(=O)Nc1ccc(N)cn1

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 3/20 0.50
HDAC1 Q13547 1/20 0.47
MAPKAPK2 P49137 6/20 0.44
GSK3B P49841 1/20 0.44
DYRK1A Q13627 1/20 0.44
NAMPT P43490 2/20 0.42
GRIN2B Q13224 1/20 0.42
MAP4K4 O95819 1/20 0.41
BCL2 P10415 1/20 0.41
ATR Q13535 1/20 0.41
MAPT P10636 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15986887 0.86 PTGS1 (0.44) PTGS1HDAC1MAPKAPK2GSK3BDYRK1A
SCHEMBL7908261 0.85 GAA (0.45) PTGS1HDAC1MAPKAPK2GSK3BDYRK1A
SCHEMBL31165993 0.85 GAA (0.45) PTGS1HDAC1MAPKAPK2GSK3BDYRK1A
SCHEMBL13403361 0.83 PTGS1 (0.51) PTGS1MAPTRAB9A
SCHEMBL6609814 0.83 NAMPT (0.52) HDAC1MAPKAPK2GSK3BDYRK1ANAMPT
SCHEMBL1126145 0.83 RAB9A (0.62) GSK3BDYRK1AMAPTRAB9A
SCHEMBL851343 0.83 DEGS1 (0.56) GSK3BDYRK1ANAMPTGRIN2B
SCHEMBL5734042 0.82 NNMT (0.58) HDAC1GSK3BDYRK1ANAMPTGRIN2B
SCHEMBL8362974 0.81 HDAC1 (0.53) HDAC1MAPKAPK2GSK3BDYRK1ANAMPT
SCHEMBL4398253 0.81 GSK3B (0.44) HDAC1MAPKAPK2GSK3BDYRK1ANAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 150 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4334298-B1 UREA DERIVATIVES WHICH CAN BE USED TO TREAT CANCER SCORPION THERAPEUTICS INC (US) 2026-02-18 EP disclosed
EP-4676923-A1 BIARYLAMIDE DERIVATIVES AND THEIR USE AS PKMYT1 INHIBITORS Cancer Research Technology Limited (GB) 2026-01-14 EP disclosed
WO-2025229624-A2 NEW CD38 INHIBITORS NAPA THERAPEUTICS LIMITED (GB) 2025-11-06 WO disclosed
WO-2025226545-A1 MODULATORS OF MITOCHONDRIAL DNA REPLICATION PRETZEL THERAPEUTICS, INC. (US) 2025-10-30 WO disclosed
US-20250250259-A1 METHODS FOR TREATING CANCER SCORPION THERAPEUTICS, INC. 2025-08-07 US disclosed
WO-2025108234-A1 COMPOUND, PREPARATION METHOD THEREFOR, AND USE THEREOF 四川科伦药物研究院有限公司 2025-05-30 WO disclosed
US-12312341-B2 Methods for treating cancer SCORPION THERAPEUTICS, INC. (US) 2025-05-27 US disclosed
WO-2025059562-A1 SUBSTITUTED AMINOPYRIDINE COMPOUNDS AND METHODS OF TREATING DISEASE USING SAME ATAVISTIK BIO, INC. (US) 2025-03-20 WO disclosed
WO-2025059469-A1 SUBSTITUTED AMINOPYRIDINE COMPOUNDS AS AKT INHIBITORS ATAVISTIK BIO, INC. (US) 2025-03-20 WO disclosed
WO-2025059577-A1 SUBSTITUTED AMINOPYRIDINE COMPOUNDS FOR USE AS AKT1 INHIBITORS ATAVISTIK BIO, INC. (US) 2025-03-20 WO disclosed
WO-2003011872-A1 PLATELET ADP RECEPTOR INHIBITORS MILLENNIUM PHARMACEUTICALS, INC. (US) 2003-02-13 WO disclosed
US-20020077486-A1 For therapy and prophylaxis of thrombosis in a mammal ALEXION PHARMACEUTICALS, INC. 2002-06-20 US disclosed
US-20020006935-A1 1-aryl-1,8-naphthylidin-4-one derivative as type IV phosphodiesterase inhibitor DAIICHI ASUBIO PHARMA CO., LTD. (JP) 2002-01-17 US disclosed
US-6297248-B1 1-aryl-1,8-naphthylidin-4-one derivative as type IV phosphodiesterase inhibitor SUNTORY LIMITED (JP) 2001-10-02 US disclosed
US-6268378-B1 TREATING AND PREVENTING OSTEOPOROSIS, AND INHIBITING VASCULAR RESTENOSIS, DIABETIC RETINOPATHY, MACULAR DEGENERATION, ANGIOGENESIS, ATHEROSCLEROSIS, INFLAMMATION, VIRAL DISEASE, AND TUMOR GROWTH. MERCK & CO., INC. 2001-07-31 US disclosed
CN-1284955-A Integrin receptor antagonists MERCK & CO INC (US) 2001-02-21 CN disclosed
US-6066648-A USEFUL IN INHIBITING BONE RESORPTION, TREATING AND PREVENTING OSTEOPOROSIS, AND INHIBITING VASCULAR RESTENOSIS, DIABETIC RETINOPATHY, MACULAR DEGENERATION, ANGIOGENESIS, ATHEROSCLEROSIS, INFLAMMATION, VIRAL DISEASE, AND TUMOR GROWTH MERCK & CO., INC. (US) 2000-05-23 US disclosed
US-6017926-A Integrin receptor antagonists MERCK & CO., INC. (US) 2000-01-25 US disclosed
EP-0958297-A1 1-ARYL-1,8-NAPHTHYLIDIN-4-ONE DERIVATIVE AS TYPE IV PHOSPHODIESTERASE INHIBITOR SUNTORY LIMITED (JP) 1999-11-24 EP disclosed
WO-1999007704-A1 1-ARYL-1,8-NAPHTHYLIDIN-4-ONE DERIVATIVE AS TYPE IV PHOSPHODIESTERASE INHIBITOR SUNTORY LIMITED (JP) 1999-02-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12312341-B2 Methods for treating cancer PIK3CA, PTEN, BRCA1 PTGS1 1077/4885HDAC1 398/4885MAPKAPK2 337/4885
US-20020077486-A1 For therapy and prophylaxis of thrombosis in a mammal PIGS, TBXA2R, GP6 PTGS1 231/4885HDAC1 1801/4885MAPKAPK2 3141/4885
US-20020006935-A1 1-aryl-1,8-naphthylidin-4-one derivative as type IV phosphodiesterase inhibitor PDE3A, PDE5A, PDE3B PTGS1 250/4885HDAC1 77/4885MAPKAPK2 2907/4885
US-20250250259-A1 METHODS FOR TREATING CANCER PIK3CA, PTEN, BRCA1 PTGS1 1077/4885HDAC1 398/4885MAPKAPK2 337/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.