SCHEMBL5633729

SCHEMBL5633729

CC(=O)N1CCN(CC#N)CC1

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.52
CYP1A2 P05177 2/20 0.46
TDP1 Q9NUW8 1/20 0.46
HRH3 Q9Y5N1 2/20 0.44
ALDH1A1 P00352 3/20 0.44
SMN1; SMN2 Q16637 1/20 0.43
RECQL P46063 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.39
KDM4E B2RXH2 3/20 0.39
DRD3 P35462 1/20 0.38
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
CYP2C9 P11712 1/20 0.38
TSHR P16473 1/20 0.38
ATM Q13315 1/20 0.37
MAPT P10636 1/20 0.37
CYP2D6 P10635 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28005050 0.81 ALDH1A1 (0.36) PIK3CDALDH1A1L3MBTL1KDM4EMEN1
SCHEMBL739637 0.81 PIK3CD (0.53) PIK3CDCYP1A2TDP1HRH3ALDH1A1
SCHEMBL3978576 0.80 ALDH1A1 (0.61) PIK3CDCYP1A2TDP1HRH3ALDH1A1
SCHEMBL299361 0.79 PIK3CD (0.52) PIK3CDCYP1A2TDP1HRH3ALDH1A1
SCHEMBL3230973 0.79 MCL1 (0.34) PIK3CDALDH1A1L3MBTL1KDM4EMEN1
SCHEMBL18702124 0.79 KMT2A (0.39) ALDH1A1L3MBTL1KDM4EMEN1KMT2A
SCHEMBL14979200 0.78 PIK3CD (0.50) PIK3CDCYP1A2TDP1HRH3SMN1; SMN2
SCHEMBL926026 0.77 TSHR (0.53) TDP1HRH3ALDH1A1SMN1; SMN2RECQL
SCHEMBL2576487 0.76 ALDH1A1 (0.50) ALDH1A1SMN1; SMN2MAPT
SCHEMBL7137154 0.76 ALDH1A1 (0.50) ALDH1A1SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170107202-A1 COMPOUNDS USEFUL AS IMMUNOMODULATORS BRISTOL-MYERS SQUIBB COMPANY 2017-04-20 US disclosed
WO-2017066227-A1 COMPOUNDS USEFUL AS IMMUNOMODULATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2017-04-20 WO disclosed
US-20170096435-A1 SEPIAPTERIN REDUCTASE INHIBITORS MAX-PLANCK-GESELLSCHAFT ZUR FOERDERUNG DER WISSENSCHAFTEN E.V. (DE) 2017-04-06 US disclosed
US-20080200433-A1 Molecular Chaperone Function Regulator MITSUBISHI TANABE PHARMA CORPORATION (JP) 2008-08-21 US disclosed
US-20070265260-A1 Quinazoline derivatives MITSUBISHI TANABE PHARMA CORPORATION (JP) 2007-11-15 US disclosed
US-7294629-B2 Quinazoline derivatives MITSUBISHI PHARMA CORPORATION (JP) 2007-11-13 US disclosed
US-7217714-B1 CCR5 modulators AGOURON PHARMACEUTICALS, INC. (US) 2007-05-15 US disclosed
US-7217714-B1 CCR5 modulators AGOURON PHARMACEUTICALS, INC. (US) 2007-05-15 US disclosed
US-7217714-B1 CCR5 modulators AGOURON PHARMACEUTICALS, INC. (US) 2007-05-15 US disclosed
CN-1150192-C Piperidines as CCR5 modulators 2004-05-19 CN disclosed
CN-1331691-A Piperidines as CCR5 modulators PFIZER LTD (US) 2002-01-16 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170096435-A1 SEPIAPTERIN REDUCTASE INHIBITORS SPR, QDPR, SRR PIK3CD 4869/4885CYP1A2 456/4885TDP1 1662/4885
US-20070265260-A1 Quinazoline derivatives TYK2, ROR1, JAK1 PIK3CD 633/4885CYP1A2 2781/4885TDP1 1537/4885
US-20170107202-A1 COMPOUNDS USEFUL AS IMMUNOMODULATORS CD74, HLA-DRB1, CD47 PIK3CD 1451/4885CYP1A2 3356/4885TDP1 2535/4885
US-20080200433-A1 Molecular Chaperone Function Regulator HSPBP1, HSF1, HSPH1 PIK3CD 3696/4885CYP1A2 4023/4885TDP1 2597/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.