SCHEMBL5645150

SCHEMBL5645150

Cc1ccccc1Pc1ccccc1Pc1ccccc1C

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.50
ACHE P22303 3/20 0.50
ALDH1A1 P00352 4/20 0.39
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
CA7 P43166 2/20 0.39
CA9 Q16790 2/20 0.39
CYP3A4 P08684 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
CYP1A2 P05177 2/20 0.36
CYP2A6 P11509 2/20 0.36
MAPT P10636 2/20 0.33
HTT P42858 1/20 0.33
LMNA P02545 1/20 0.33
ALOX12 P18054 1/20 0.33
ESR1 P03372 1/20 0.33
TAAR1 Q96RJ0 1/20 0.32
HSD17B10 Q99714 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL146928 0.97 TSHR (0.53) TSHRACHEALDH1A1CA1CA2
SCHEMBL1304780 0.94 TSHR (0.50) TSHRACHEALDH1A1CA1CA2
SCHEMBL31457202 0.94 TSHR (0.50) TSHRACHEALDH1A1CA1CA2
Hydrochloric Acid SCHEMBL541709 0.94 TSHR (0.50) TSHRACHEALDH1A1CA1CA2
SCHEMBL29083664 0.94 TSHR (0.50) TSHRACHEALDH1A1CA1CA2
Hydrochloric Acid SCHEMBL29042332 0.92 TSHR (0.47) TSHRACHEALDH1A1CA1CA2
Hydrochloric Acid SCHEMBL3223494 0.92 TSHR (0.47) TSHRACHEALDH1A1CA1CA2
Bromide SCHEMBL29042359 0.92 TSHR (0.47) TSHRACHEALDH1A1CA1CA2
Propane SCHEMBL29069359 0.89 TSHR (0.45) TSHRACHEALDH1A1CA1CA2
SCHEMBL3632065 0.87 ACHE (0.43) TSHRACHEALDH1A1CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006057904-A1 STEREOSELECTIVE PREPARATION OF 4-ARYL PIPERIDINE AMIDES BY ASYMMETRIC HYDROGENATION OF A PROCHIRAL ENAMIDE AND INTERMEDIATES OF THIS PROCESS MERCK & CO., INC. (US) 2006-06-01 WO claimed
US-7230134-B2 Method for the production of amines by reductive amination of carbonyl compounds under transfer-hydrogenation conditions DEGUSSA AG (DE) 2007-06-12 US disclosed
WO-2006057904-A1 STEREOSELECTIVE PREPARATION OF 4-ARYL PIPERIDINE AMIDES BY ASYMMETRIC HYDROGENATION OF A PROCHIRAL ENAMIDE AND INTERMEDIATES OF THIS PROCESS MERCK & CO., INC. (US) 2006-06-01 WO disclosed
US-20040267051-A1 Method for the production of amines by reductive amination of carbonyl compounds under transfer-hydrogenation conditions EVONIK DEGUSSA GMBH (DE) 2004-12-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040267051-A1 Method for the production of amines by reductive amination of carbonyl compounds under transfer-hydrogenation conditions HNMT, AADAT, ADH5 TSHR 2166/4885ACHE 1456/4885ALDH1A1 248/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.