SCHEMBL5659286

SCHEMBL5659286

COc1ccccc1N(CCCN1CCN(c2ccc(Cl)nn2)CC1)C(=O)O

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.52
LMNA P02545 1/20 0.52
HTR4 Q13639 1/20 0.49
DRD2 P14416 8/20 0.44
HTR2A P28223 2/20 0.42
KDM4E B2RXH2 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
DRD4 P21917 1/20 0.41
DRD3 P35462 1/20 0.41
OPRM1 P35372 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HTR1A P08908 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5656932 0.91 OPRM1 (0.46) ALDH1A1LMNAHTR4DRD2HTR2A
SCHEMBL5656321 0.87 HTR4 (0.49) ALDH1A1HTR4DRD2HTR2AKDM4E
SCHEMBL5659379 0.85 LMNA (0.44) ALDH1A1LMNAHTR4DRD4OPRM1
SCHEMBL5656351 0.84 HTR1A (0.57) ALDH1A1DRD2HTR2AKDM4ESMN1; SMN2
SCHEMBL5654725 0.83 DRD2 (0.55) ALDH1A1DRD2HTR2AKDM4ETDP1
SCHEMBL5657861 0.83 OPRM1 (0.55) ALDH1A1HTR4DRD2HTR2AKDM4E
SCHEMBL5655983 0.82 MAPT (0.53) DRD2HTR2ADRD4DRD3OPRM1
SCHEMBL5659495 0.82 OPRM1 (0.50) ALDH1A1DRD2HTR2AKDM4ETDP1
SCHEMBL5657431 0.82 LMNA (0.53) ALDH1A1LMNAHTR4DRD2HTR2A
SCHEMBL5655837 0.82 DRD2 (0.63) ALDH1A1DRD2HTR2AKDM4ETDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7238693-B2 Aryl carbamate derivatives, preparation and use thereof CEREP (FR) 2007-07-03 US disclosed
US-20040058933-A1 Aryl carbamate derivatives, preperation and use thereof CEREP (FR) 2004-03-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040058933-A1 Aryl carbamate derivatives, preperation and use thereof HTR4, HTR5A, HTR3C ALDH1A1 1018/4885LMNA 1137/4885HTR4 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.