SCHEMBL5689270

SCHEMBL5689270

COc1ccc(-c2ccccc2)cc1C(O)c1c[nH]cn1

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CTSA P10619 8/20 0.44
DHFR P00374 2/20 0.38
AAK1 Q2M2I8 1/20 0.38
KIT P10721 1/20 0.38
IDO1 P14902 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.36
ACHE P22303 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11051393 0.84 SMN1; SMN2 (0.45) IDO1SMN1; SMN2ACHE
SCHEMBL6929116 0.79 CASR (0.39) CTSAAAK1KITIDO1SMN1; SMN2
SCHEMBL6266844 0.71 CYP2D6 (0.46) CTSADHFR
SCHEMBL7159560 0.70 ROCK2 (0.38) SMN1; SMN2ACHE
SCHEMBL7159601 0.70 ACHE (0.38) SMN1; SMN2ACHE
SCHEMBL7098179 0.70 ALDH1A1 (0.38) KITSMN1; SMN2ACHE
SCHEMBL5688780 0.70 RAB9A (0.47) CTSAAAK1KIT
SCHEMBL21376221 0.70 DHFR (0.48) CTSADHFR
SCHEMBL5688342 0.69 CYP17A1 (0.44) CTSAAAK1KITIDO1
SCHEMBL11045849 0.69 TSHR (0.34) SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1227086-B1 1-SUBSTITUTED PHENYL-1-(1H-IMIDAZOL-4-YL) ALCOHOLS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2006-03-29 EP disclosed
US-6518257-B1 1-substituted phenyl-1-(1h-imidazol-4-yl) alcohols, process for producing the same and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-02-11 US disclosed
EP-1227086-A1 1-SUBSTITUTED PHENYL-1-(1H-IMIDAZOL-4-YL) ALCOHOLS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-07-31 EP disclosed