SCHEMBL5690356

SCHEMBL5690356

COC(=O)[C@H](Cc1ccc(NC(=O)C2CCN(C(=O)OCc3ccccc3)CC2)cc1)N(C(=O)C1CNCCN1C(=O)OCc1ccccc1)S(=O)(=O)c1ccc(C)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 9/20 0.48
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HTT P42858 1/20 0.41
F13A1 P00488 1/20 0.39
TGM2 P21980 1/20 0.39
TGM1 P22735 1/20 0.39
KDM4E B2RXH2 1/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
TRPV1 Q8NER1 1/20 0.39
ALDH1A1 P00352 2/20 0.39
GAA P10253 1/20 0.39
MMP1 P03956 1/20 0.39
MMP2 P08253 1/20 0.39
MMP3 P08254 1/20 0.39
MMP7 P09237 1/20 0.39
MMP9 P14780 1/20 0.39
MMP8 P22894 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5690403 0.95 ENPP2 (0.47) ENPP2NPC1RAB9ASMN1; SMN2HTT
SCHEMBL5690361 0.75 ENPP3 (0.39) ENPP2SMN1; SMN2HTTLMNAMAPT
SCHEMBL7970301 0.74 PTPN2 (0.44) NPC1RAB9ALMNAMAPTTRPV1
SCHEMBL5690604 0.74 ENPP2 (0.48) ENPP2NPC1RAB9ASMN1; SMN2HTT
SCHEMBL5690337 0.72 ENPP2 (0.49) ENPP2NPC1RAB9ASMN1; SMN2HTT
SCHEMBL5691009 0.72 MAPT (0.40) ENPP2SMN1; SMN2HTTLMNAMAPT
SCHEMBL5691183 0.72 ITGB1 (0.60) ENPP2ALDH1A1MMP1MMP2MMP3
SCHEMBL5690873 0.72 ITGB1 (0.60) ENPP2ALDH1A1MMP1MMP2MMP3
SCHEMBL5690759 0.72 TRPV1 (0.41) ENPP2SMN1; SMN2HTTLMNAMAPT
Hydrochloric Acid SCHEMBL5681091 0.71 ENPP2 (0.66) ENPP2NPC1RAB9ASMN1; SMN2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001974-B1 4-AMINO-PHENYLALANINE TYPE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARM INC (US) 2006-05-24 EP claimed
EP-1001974-B1 4-AMINO-PHENYLALANINE TYPE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARM INC (US) 2006-05-24 EP disclosed