SCHEMBL5696188

SCHEMBL5696188

Oc1cccc(C2NC(=S)Nc3ccc(Br)cc32)c1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.50
GUSB P08236 1/20 0.45
BCHE P06276 1/20 0.37
ACHE P22303 1/20 0.37
KIF11 P52732 5/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
DRD2 P14416 1/20 0.35
DRD3 P35462 1/20 0.35
KDM1A O60341 1/20 0.35
TP53 P04637 2/20 0.35
MAPK1 P28482 1/20 0.35
HSD17B10 Q99714 1/20 0.35
GAA P10253 1/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29857451 1.00 DHFR (0.50) DHFRGUSBBCHEACHEKIF11
SCHEMBL5696173 0.84 DHFR (0.50) DHFRGUSBKIF11MEN1KMT2A
SCHEMBL5696233 0.83 DHFR (0.54) DHFRGUSBKIF11MEN1KMT2A
SCHEMBL29357488 0.83 DHFR (0.54) DHFRGUSBKIF11MEN1KMT2A
SCHEMBL5696249 0.77 DHFR (0.51) DHFRGUSBKIF11
SCHEMBL5176445 0.77 DHFR (0.51) DHFRGUSBKIF11MAPK1HSD17B10
SCHEMBL5176914 0.73 LMNA (0.41) MEN1KMT2ATP53GAALMNA
SCHEMBL9701173 0.73 DHFR (0.62) DHFRGUSBKIF11MAPK1HSD17B10
SCHEMBL5696167 0.72 DHFR (0.57) DHFRGUSBBCHEACHEKIF11
SCHEMBL5696196 0.69 DHFR (0.51) DHFRGUSBKIF11MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1655289-A1 Quinazoline derivatives, process for their preparation, their use as antimitotics and pharmaceutical compositions comprising said derivatives EMBL (DE) 2006-05-10 EP disclosed