SCHEMBL5696173

SCHEMBL5696173

Oc1cccc(C2NC(=S)Nc3ccc(Cl)cc32)c1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.50
GUSB P08236 1/20 0.45
HTR2A P28223 2/20 0.40
HTR2C P28335 2/20 0.40
TSHR P16473 1/20 0.38
ATM Q13315 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
TRPM4 Q8TD43 1/20 0.36
TRPM5 Q9NZQ8 1/20 0.36
KIF11 P52732 7/20 0.36
ALDH1A1 P00352 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.35
ALOX12 P18054 1/20 0.34
HTT P42858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5696249 0.91 DHFR (0.51) DHFRGUSBHTR2AHTR2CTSHR
SCHEMBL5205016 0.85 ALDH1A1 (0.46) TSHRATMMEN1KMT2ATRPM4
SCHEMBL5696188 0.84 DHFR (0.50) DHFRGUSBMEN1KMT2AKIF11
SCHEMBL29857451 0.84 DHFR (0.50) DHFRGUSBMEN1KMT2AKIF11
SCHEMBL5696233 0.83 DHFR (0.54) DHFRGUSBMEN1KMT2AKIF11
SCHEMBL29357488 0.83 DHFR (0.54) DHFRGUSBMEN1KMT2AKIF11
SCHEMBL5176445 0.77 DHFR (0.51) DHFRGUSBHTR2AHTR2CKIF11
SCHEMBL5177579 0.76 ALDH1A1 (0.46) DHFRGUSBHTR2AHTR2CMEN1
SCHEMBL5177430 0.75 MAPT (0.50) HTR2AHTR2CTSHRATMMEN1
SCHEMBL5696272 0.73 CHRM1 (0.42) HTR2AHTR2CTSHRKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1655289-A1 Quinazoline derivatives, process for their preparation, their use as antimitotics and pharmaceutical compositions comprising said derivatives EMBL (DE) 2006-05-10 EP disclosed