SCHEMBL5696249

SCHEMBL5696249

Oc1cccc(C2NC(=S)Nc3cc(Cl)ccc32)c1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.51
GUSB P08236 1/20 0.46
HTR2A P28223 2/20 0.44
HTR2C P28335 2/20 0.44
TSHR P16473 1/20 0.39
KIF11 P52732 9/20 0.38
ALDH1A1 P00352 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HTT P42858 1/20 0.35
PDE4A P27815 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5696173 0.91 DHFR (0.50) DHFRGUSBHTR2AHTR2CTSHR
SCHEMBL5177579 0.86 ALDH1A1 (0.46) DHFRGUSBHTR2AHTR2CKIF11
SCHEMBL5696233 0.85 DHFR (0.54) DHFRGUSBKIF11ALDH1A1HTT
SCHEMBL29357488 0.85 DHFR (0.54) DHFRGUSBKIF11ALDH1A1HTT
SCHEMBL5176445 0.84 DHFR (0.51) DHFRGUSBHTR2AHTR2CKIF11
SCHEMBL5696188 0.77 DHFR (0.50) DHFRGUSBKIF11
SCHEMBL29857451 0.77 DHFR (0.50) DHFRGUSBKIF11
SCHEMBL5205016 0.74 ALDH1A1 (0.46) TSHRKIF11ALDH1A1
SCHEMBL9701173 0.74 DHFR (0.62) DHFRGUSBKIF11ALDH1A1SMN1; SMN2
SCHEMBL5696167 0.73 DHFR (0.57) DHFRGUSBKIF11ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1655289-A1 Quinazoline derivatives, process for their preparation, their use as antimitotics and pharmaceutical compositions comprising said derivatives EMBL (DE) 2006-05-10 EP disclosed