SCHEMBL569815

SCHEMBL569815

CC(C)(C)N1CC(O)(c2ccc([Si](C)(C)C)cc2)C1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.37
NR1H2 P55055 1/20 0.34
NR1H3 Q13133 1/20 0.34
OPRM1 P35372 2/20 0.32
GRIN2D O15399 1/20 0.32
GRIN3B O60391 1/20 0.32
CHRM2 P08172 1/20 0.32
CHRM1 P11229 1/20 0.32
GRIN1 Q05586 1/20 0.32
KCNH2 Q12809 1/20 0.32
GRIN2A Q12879 1/20 0.32
GRIN2B Q13224 1/20 0.32
GRIN2C Q14957 1/20 0.32
GRIN3A Q8TCU5 1/20 0.32
OPRD1 P41143 1/20 0.31
OPRK1 P41145 1/20 0.31
OPRL1 P41146 1/20 0.31
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15543215 0.79 OPRM1 (0.43) ALDH1A1OPRM1CHRM1KCNH2OPRD1
SCHEMBL18115648 0.78 ALDH1A1 (0.58) ALDH1A1OPRM1GRIN2DGRIN3BCHRM2
SCHEMBL23748773 0.76 OPRM1 (0.37) ALDH1A1OPRM1GRIN2DGRIN3BGRIN1
SCHEMBL24421814 0.76 ALDH1A1 (0.37) ALDH1A1OPRM1GRIN2DGRIN3BCHRM2
SCHEMBL15544188 0.75 OPRM1 (0.47) ALDH1A1OPRM1GRIN2BOPRD1OPRK1
SCHEMBL20341691 0.71
SCHEMBL24422423 0.71 ALDH1A1 (0.33) ALDH1A1KCNH2
SCHEMBL15212418 0.71 LMNA (0.34) ALDH1A1MAPT
SCHEMBL23748779 0.67 CCR1 (0.42) ALDH1A1OPRM1GRIN2DGRIN3BCHRM2
SCHEMBL16936786 0.67 MAPT (0.51) ALDH1A1OPRM1OPRD1OPRK1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2601190-A1 ISOXAZOLINE DERIVATIVES AS ANTIPARASITIC AGENTS AH USA 42 LLC (US) 2013-06-12 EP disclosed
WO-2012017359-A1 ISOXAZOLINE DERIVATIVES AS ANTIPARASITIC AGENTS PFIZER INC. (US) 2012-02-09 WO disclosed