Eprobemide

Eprobemide

SCHEMBL570896

O=C(NCCCN1CCOCC1)c1ccc(Cl)cc1

nearest known ligand 0.86

Full drug profile on Sugi Atlas →

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.85
HTR1A P08908 1/20 0.85
MAOA P21397 1/20 0.85
MAOB P27338 1/20 0.85
KCNH2 Q12809 1/20 0.85
CD274 Q9NZQ7 1/20 0.85
TSHR P16473 1/20 0.76
MEN1 O00255 1/20 0.76
KMT2A Q03164 1/20 0.76
KDM4E B2RXH2 1/20 0.72
SMN1; SMN2 Q16637 1/20 0.72
EPHX2 P34913 1/20 0.72
TMEM97 Q5BJF2 1/20 0.64
SIGMAR1 Q99720 1/20 0.64
CYP2D6 P10635 1/20 0.63
CYP2C9 P11712 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Eprobemide SCHEMBL10495496 0.99 ALDH1A1 (0.82) ALDH1A1HTR1AMAOAMAOBKCNH2
Moclobemide SCHEMBL3408310 0.92 CD274 (1.00) ALDH1A1HTR1AMAOAMAOBKCNH2
Moclobemide SCHEMBL49708 0.92 CD274 (1.00) ALDH1A1HTR1AMAOAMAOBKCNH2
Moclobemide SCHEMBL11475483 0.90 CD274 (0.97) ALDH1A1HTR1AMAOAMAOBKCNH2
SCHEMBL10756632 0.90 TMEM97 (0.72) ALDH1A1HTR1AMAOAMAOBKCNH2
SCHEMBL2249600 0.88 TSHR (0.74) ALDH1A1HTR1AMAOAMAOBKCNH2
SCHEMBL12459935 0.86 CD274 (0.79) ALDH1A1HTR1AMAOAMAOBKCNH2
SCHEMBL763452 0.86 HTT (0.78) ALDH1A1HTR1AMAOAMAOBKCNH2
SCHEMBL1382764 0.86 SMN1; SMN2 (0.95) ALDH1A1CD274TSHRKDM4ESMN1; SMN2
SCHEMBL12089972 0.86 LMNA (0.83) ALDH1A1HTR1AMAOAMAOBKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 682 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250339403-A1 Tryptamine Formulations and Uses Thereof Natural MedTech Pty Ltd (AU) 2025-11-06 US claimed
EP-4633638-A1 TREATMENT OF PSYCHOLOGICAL FACTORS AFFECTING OTHER MEDICAL CONDITIONS (PFAOMC) Luminous Mind Inc. (US) 2025-10-22 EP claimed
EP-4615444-A1 TRYPTAMINE FORMULATIONS AND USES THEREOF Natural Medtech Pty Ltd (AU) 2025-09-17 EP claimed
EP-4479032-A1 NEUROACTIVE STEROIDS FOR TREATMENT OF CNS-RELATED DISORDERS Sage Therapeutics, Inc. (US) 2024-12-25 EP claimed
WO-2024130044-A1 TREATMENT OF PSYCHOLOGICAL FACTORS AFFECTING OTHER MEDICAL CONDITIONS (PFAOMC) LUMINOUS MIND INC. (US) 2024-06-20 WO claimed
WO-2024098098-A1 TRYPTAMINE FORMULATIONS AND USES THEREOF Natural MedTech Pty Ltd (AU) 2024-05-16 WO claimed
US-20230390220-A1 MONOAMINE OXIDASE BLOCKADE THERAPY FOR TREATING CANCER THROUGH REGULATING ANTITUMOR T CELL IMMUNITY THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-12-07 US claimed
US-20230391871-A1 MONOAMINE OXIDASE BLOCKADE THERAPY FOR TREATING CANCER THROUGH REGULATING TUMOR ASSOCIATED MACROPHAGES (TAMS) THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-12-07 US claimed
US-20230381168-A1 ADJUNCTIVE THERAPY FOR DEPRESSION ANEUROTECH BV (BE) 2023-11-30 US claimed
EP-4277612-A1 COMBINATION OF AN ANTIDEPRESSANT AND DEXTROMETHORPHAN FOR NEUROPSYCHIATRIC CONDITIONS Antecip Bioventures II LLC (US) 2023-11-22 EP claimed
US-7053080-B2 Methods and therapeutic combinations for the treatment of obesity using sterol absorption inhibitors SCHERING CORPORATION (US) 2006-05-30 US claimed
US-20060009399-A1 Methods and therapeutic combinations for the treatment of obesity using sterol absorption inhibitors DAVIS HARRY R 2006-01-12 US claimed
US-20030119428-A1 Methods and therapeutic combinations for the treatment of obesity using sterol absorption inhibitors SCHERING CORPORATION 2003-06-26 US claimed
CN-1370067-A Use of monoamine oxidase inhibitors for manufacture of drugs intended for treatment of obesity SANOFI SYNTHELABO (FR) 2002-09-18 CN claimed
EP-1210080-A2 USE OF MONOAMINE OXIDASE INHIBITORS FOR THE MANUFACTURE OF DRUGS INTENDED FOR THE TREATMENT OF OBESITY Sanofi-Aventis (FR) 2002-06-05 EP claimed
EP-1150715-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING NICOTINE OR A LIGAND OF NICOTINE RECEPTORS AND A MONAMINE OXYDASE INHIBITOR AND THEIR USE FOR TREATING TOBACCO WITHDRAWAL SYMPTOMS SANOFI-SYNTHELABO (FR) 2001-11-07 EP claimed
EP-1078632-A1 Use of monoamine oxydase inhibitors for the manufacture of drugs intended for the treatment of obesity SANOFI-SYNTHELABO (FR) 2001-02-28 EP claimed
WO-2001012176-A2 USE OF MONOAMINE OXIDASE INHIBITORS FOR THE MANUFACTURE OF DRUGS INTENDED FOR THE TREATMENT OF OBESITY SANOFI-SYNTHELABO (FR) 2001-02-22 WO claimed
WO-2000045846-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING NICOTINE OR A LIGAND OF NICOTINE RECEPTORS AND A MONAMINE OXYDASE INHIBITOR AND THEIR USE FOR TREATING TOBACCO WITHDRAWAL SYMPTOMS SANOFI-SYNTHELABO (FR) 2000-08-10 WO claimed
WO-1999013879-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING A MONOAMINE OXYDASE INHIBITOR AND THEIR USE IN THERAPY SANOFI-SYNTHELABO (FR) 1999-03-25 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060009399-A1 Methods and therapeutic combinations for the treatment of obesity using sterol absorption inhibitors NPC1L1, SLC10A2, SLC10A1 ALDH1A1 1403/4885HTR1A 2184/4885MAOA 2912/4885
US-20230381168-A1 ADJUNCTIVE THERAPY FOR DEPRESSION HTR2A, HTR3B, HTR5A ALDH1A1 1086/4885HTR1A 6/4885MAOA 183/4885
US-20250339403-A1 Tryptamine Formulations and Uses Thereof MAOA, MAOB, TPH1 ALDH1A1 636/4885HTR1A 15/4885MAOA 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.