SCHEMBL571200

SCHEMBL571200

C=C1C[C@@H](C(=O)O)N(C(=O)OC(C)(C)C)C1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.37
PTPN1 P18031 2/20 0.37
CHRM2 P08172 1/20 0.35
CHRM1 P11229 1/20 0.35
CHRM3 P20309 1/20 0.35
NPC1 O15118 1/20 0.34
GPR119 Q8TDV5 1/20 0.34
HDAC8 Q9BY41 2/20 0.34
LMNA P02545 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
USP2 O75604 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL206317 1.00 HSD17B10 (0.42) HSD17B10SMN1; SMN2PTPN1CHRM2CHRM1
SCHEMBL22364678 0.89 HSD17B10 (0.38) HSD17B10SMN1; SMN2PTPN1CHRM2CHRM1
SCHEMBL2009986 0.87 PTPN1 (0.42) HSD17B10SMN1; SMN2PTPN1CHRM2CHRM1
SCHEMBL2009984 0.87 PTPN1 (0.42) HSD17B10SMN1; SMN2PTPN1CHRM2CHRM1
SCHEMBL20054308 0.87 CHRM2 (0.38) HSD17B10SMN1; SMN2PTPN1CHRM2CHRM1
SCHEMBL15116703 0.87 CHRM2 (0.38) HSD17B10SMN1; SMN2PTPN1CHRM2CHRM1
SCHEMBL16824577 0.86 HSD17B10 (0.47) HSD17B10SMN1; SMN2NPC1GPR119LMNA
SCHEMBL16824578 0.86 HSD17B10 (0.47) HSD17B10SMN1; SMN2NPC1GPR119LMNA
SCHEMBL239567 0.86 PTPN1 (0.36) HSD17B10PTPN1CHRM2CHRM1CHRM3
SCHEMBL239566 0.86 PTPN1 (0.36) HSD17B10PTPN1CHRM2CHRM1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 442 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118684615-A Synthesis method of difluoro cyclobutane proline and derivative thereof 吉尔多肽生物制药(大连市)有限公司 2024-09-24 CN claimed
US-20250353833-A1 DPP9 BINDING COMPOUNDS UNIV ANTWERPEN (BE) 2025-11-20 US disclosed
US-20250346585-A1 PHARMACEUTICAL COMPOUNDS FOR THE TREATMENT OF COMPLEMENT MEDIATED DISORDERS ALEXION PHARMACEUTICALS, INC. (US) 2025-11-13 US disclosed
EP-4640684-A1 KRAS G12D INHIBITORS AND USES THEREOF Abbisko Therapeutics Co., Ltd. (CN) 2025-10-29 EP disclosed
US-20250281424-A1 SMALL MOLECULE ANTAGONISTS OF PF4 ZHOU YUHANG (US) 2025-09-11 US disclosed
CN-119894891-A KRAS G12D inhibitor and application thereof 上海和誉生物医药科技有限公司 2025-04-25 CN disclosed
WO-2024235121-A1 FUSED RING COMPOUND AND PREPARATION METHOD THEREFOR AND USE THEREOF 四川科伦博泰生物医药股份有限公司 2024-11-21 WO disclosed
US-12139497-B2 Aryl, heteroaryl, and heterocyclic compounds for treatment of medical disorders ACHILLION PHARMACEUTICALS, INC. (US) 2024-11-12 US disclosed
US-20240317748-A1 CARBONYL SUBSTITUTED DIAZASPIRO COMPOUNDS AND ITS USE BIONOVA PHARMACEUTICALS LTD. (KY) 2024-09-26 US disclosed
CN-118684615-A Synthesis method of difluoro cyclobutane proline and derivative thereof 吉尔多肽生物制药(大连市)有限公司 2024-09-24 CN disclosed
US-20030171309-A1 Pharmaceutically active pyrrolidine derivatives as bax inhibitors MERCK SERONO SA (CH) 2003-09-11 US disclosed
CN-1419541-A Pharmaceutically active pyrrolidine derivatives as BAX inhibitors APPLIED RES SYSTEMS AKS HOLDIN (NL) 2003-05-21 CN disclosed
EP-1303486-A1 PYRROLIDINE DERIVATIVES AS METALLOPROTEASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2003-04-23 EP disclosed
EP-1268419-A1 PYRROLIDINE DERIVATIVES USEFUL AS BAX INHIBITORS Applied Research Systems ARS Holding N.V. (AN) 2003-01-02 EP disclosed
EP-1268418-A1 PHARMACEUTICALLY ACTIVE PYRROLIDINE DERIVATIVES AS BAX INHIBITORS Applied Research Systems ARS Holding N.V. (AN) 2003-01-02 EP disclosed
US-20020040146-A1 Pyrrolidine derivatives F. HOFFMANN-LA ROCHE AG, A SWISS COMPANY (CH) 2002-04-04 US disclosed
WO-2002008185-A1 PYRROLIDINE DERIVATIVES AS METALLOPROTEASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2002-01-31 WO disclosed
WO-2001074769-A1 PHARMACEUTICALLY ACTIVE PYRROLIDINE DERIVATIVES AS BAX INHIBITORS APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2001-10-11 WO disclosed
WO-2001072705-A1 PHARMACEUTICALLY ACTIVE PYRROLIDINE DERIVATIVES AS BAX INHIBITORS APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2001-10-04 WO disclosed
WO-1995004718-A1 4-METHYLENEPROLINE DERIVATIVES AS FUNGICIDES ZENECA LIMITED (GB) 1995-02-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240317748-A1 CARBONYL SUBSTITUTED DIAZASPIRO COMPOUNDS AND ITS USE SDHA, PDHA1, GLS HSD17B10 1040/4885SMN1; SMN2 498/4885PTPN1 4092/4885
US-20250281424-A1 SMALL MOLECULE ANTAGONISTS OF PF4 PF4, F12, F2 HSD17B10 1989/4885SMN1; SMN2 4700/4885PTPN1 1325/4885
US-20250346585-A1 PHARMACEUTICAL COMPOUNDS FOR THE TREATMENT OF COMPLEMENT MEDIATED DISORDERS C5, C1S, C9 HSD17B10 2484/4885SMN1; SMN2 266/4885PTPN1 3684/4885
US-20020040146-A1 Pyrrolidine derivatives PREP, PEPD, MMP3 HSD17B10 1522/4885SMN1; SMN2 3344/4885PTPN1 3435/4885
US-20250353833-A1 DPP9 BINDING COMPOUNDS DPP9, DPP7, DPP3 HSD17B10 804/4885SMN1; SMN2 4493/4885PTPN1 920/4885
US-12139497-B2 Aryl, heteroaryl, and heterocyclic compounds for treatment of medical disorders CFD, F12, F3 HSD17B10 991/4885SMN1; SMN2 2468/4885PTPN1 3140/4885
US-20030171309-A1 Pharmaceutically active pyrrolidine derivatives as bax inhibitors SUCNR1, PYCR1, GLS HSD17B10 1885/4885SMN1; SMN2 459/4885PTPN1 1229/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.