SCHEMBL5721087

SCHEMBL5721087

CNC(=O)C(CC(C)COC)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GLS O94925 2/20 0.43
CRHBP P24387 1/20 0.43
CRHR2 Q13324 1/20 0.43
ALDH1A1 P00352 4/20 0.42
HPGD P15428 2/20 0.41
GPR88 Q9GZN0 3/20 0.41
LMNA P02545 1/20 0.41
TSHR P16473 1/20 0.41
CTSS P25774 2/20 0.40
CTSK P43235 2/20 0.40
CTSL P07711 1/20 0.40
MMP1 P03956 1/20 0.40
MMP2 P08253 1/20 0.40
MMP3 P08254 1/20 0.40
MMP9 P14780 1/20 0.40
MMP14 P50281 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5196291 0.86 GLS (0.53) GLSCRHBPCRHR2ALDH1A1HPGD
Ethane SCHEMBL27961526 0.80 CTSK (0.55) CRHBPCRHR2ALDH1A1LMNACTSS
SCHEMBL2049579 0.74 ALDH1A1 (0.66) CRHBPCRHR2ALDH1A1LMNAKMT2A
SCHEMBL2721958 0.74 LMNA (0.50) GLSCRHBPCRHR2ALDH1A1GPR88
SCHEMBL9055208 0.73 ROCK2 (0.50) GLSCRHBPCRHR2ALDH1A1LMNA
SCHEMBL7504901 0.73 LMNA (0.49) CRHBPCRHR2ALDH1A1LMNA
SCHEMBL19256857 0.73 ROCK2 (0.50) GLSCRHBPCRHR2ALDH1A1LMNA
SCHEMBL819828 0.73 KMT2A (0.58) GLSALDH1A1HPGDLMNATSHR
SCHEMBL2016945 0.72 CYP2C19 (0.52) GLSALDH1A1HPGDLMNATSHR
SCHEMBL19932307 0.72 CRHBP (0.47) CRHBPCRHR2ALDH1A1LMNAMMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1682494-A4 ARALKYL AMINES AS CANNABINOID RECEPTOR MODULATORS MERCK & CO INC (US) 2006-11-08 EP disclosed
EP-1682494-A1 ARALKYL AMINES AS CANNABINOID RECEPTOR MODULATORS Merck & Co., Inc. (US) 2006-07-26 EP disclosed
WO-2005044785-A1 ARALKYL AMINES AS CANNABINOID RECEPTOR MODULATORS MERCK & CO., INC. (US) 2005-05-19 WO disclosed