SCHEMBL5737282

SCHEMBL5737282

Cc1ccc(-c2ccc(C=O)o2)cc1C

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.56
ALDH1A1 P00352 7/20 0.56
LMNA P02545 2/20 0.56
LDHA P00338 1/20 0.53
LDHB P07195 1/20 0.53
HAO1 Q9UJM8 1/20 0.53
TDP1 Q9NUW8 2/20 0.51
MAPT P10636 6/20 0.50
POLB P06746 4/20 0.50
NPC1 O15118 2/20 0.50
RAB9A P51151 2/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
HSP90AA1 P07900 1/20 0.50
HPGD P15428 3/20 0.49
TP53 P04637 1/20 0.49
SMN1; SMN2 Q16637 4/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
CYP2E1 P05181 1/20 0.46
CYP3A4 P08684 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2319080 0.85 KDM4E (0.60) KDM4EALDH1A1LMNALDHALDHB
SCHEMBL2321202 0.85 KDM4E (0.58) KDM4EALDH1A1LMNALDHALDHB
SCHEMBL7833840 0.85 ALDH1A1 (0.51) KDM4EALDH1A1LMNALDHALDHB
SCHEMBL4704691 0.85 LDHA (0.64) KDM4EALDH1A1LMNALDHALDHB
SCHEMBL2553518 0.81 LDHA (0.72) KDM4EALDH1A1LMNALDHALDHB
SCHEMBL396870 0.80 ALDH1A1 (0.80) KDM4EALDH1A1LMNALDHALDHB
SCHEMBL6589648 0.80 MAPT (0.59) KDM4EALDH1A1LMNALDHALDHB
SCHEMBL2318474 0.79 KDM4E (0.67) KDM4EALDH1A1LMNALDHALDHB
SCHEMBL10092801 0.78 ALDH1A1 (0.65) KDM4EALDH1A1LMNALDHALDHB
SCHEMBL7036878 0.78 ALDH1A1 (0.58) KDM4EALDH1A1LMNALDHALDHB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8466291-B2 1,5-dideoxy-1,5-imino-D-glucitol compounds ACADEMIA SINICA (TW) 2013-06-18 US disclosed
US-8466291-B2 1,5-dideoxy-1,5-imino-D-glucitol compounds ACADEMIA SINICA (TW) 2013-06-18 US disclosed
US-20100113519-A1 1,5-Dideoxy-1,5-imino-D-glucitol Compounds ACADEMIA SINICA (TW) 2010-05-06 US disclosed
US-20100113519-A1 1,5-Dideoxy-1,5-imino-D-glucitol Compounds ACADEMIA SINICA (TW) 2010-05-06 US disclosed
EP-1244446-B1 THROMBOPOIETIN MIMETICS SMITHKLINE BEECHAM CORP (US) 2006-11-02 EP disclosed
US-6858630-B2 Naphthimidazole derivatives and their use as thrombopoietin mimetics SMITHKLINE BEECHAM CORPORATION (US) 2005-02-22 US disclosed
US-20030083361-A1 Naphtho(1,2-d)imidazole derivatives; treating thrombocytopenia SMITHKLINE BEECHAM CORPORATION 2003-05-01 US disclosed
EP-1244446-A4 THROMBOPOIETIN MIMETICS SMITHKLINE BEECHAM CORP (US) 2003-01-08 EP disclosed
EP-1244446-A1 THROMBOPOIETIN MIMETICS SmithKline Beecham Corporation (US) 2002-10-02 EP disclosed
WO-2001039773-A1 THROMBOPOIETIN MIMETICS SMITHKLINE BEECHAM CORPORATION (US) 2001-06-07 WO disclosed
US-4123529-A TREATMENT OF ASTHMA LILLY INDUSTRIES LIMITED (GB) 1978-10-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030083361-A1 Naphtho(1,2-d)imidazole derivatives; treating thrombocytopenia MPL, THPO, TPO KDM4E 4286/4885ALDH1A1 2193/4885LMNA 3899/4885
US-20100113519-A1 1,5-Dideoxy-1,5-imino-D-glucitol Compounds HEXD, GALE, GBA1 KDM4E 3356/4885ALDH1A1 321/4885LMNA 1440/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.