SCHEMBL574089

SCHEMBL574089

CC1(C)OB(c2csc3ccccc23)OC1(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.41
LPL P06858 6/20 0.40
LIPG Q9Y5X9 6/20 0.40
CYP2A6 P11509 3/20 0.38
PKM P14618 2/20 0.36
CHRNA7 P36544 1/20 0.34
SLC6A4 P31645 1/20 0.34
HDAC3 O15379 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC7 Q8WUI4 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC10 Q969S8 1/20 0.33
HDAC11 Q96DB2 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
HDAC9 Q9UKV0 1/20 0.33
HDAC5 Q9UQL6 1/20 0.33
CRHBP P24387 1/20 0.33
CRHR2 Q13324 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28543534 0.80 CYP2A6 (0.44) MAPTCYP2A6PKMCHRNA7SLC6A4
SCHEMBL23645509 0.79 MAPT (0.37) MAPTLPLLIPGCYP2A6
SCHEMBL14727554 0.78 LPL (0.43) MAPTLPLLIPGSLC6A4KDM4E
SCHEMBL657279 0.78 MAP3K7 (0.34) LPLLIPGCYP2A6
SCHEMBL25027588 0.78 LPL (0.41) MAPTLPLLIPGALDH1A1
SCHEMBL30445860 0.78 MAP3K7 (0.34) LPLLIPGCYP2A6
SCHEMBL13927329 0.78 LPL (0.41) MAPTLPLLIPG
SCHEMBL15574699 0.78 CYP2A6 (0.41) LPLLIPGCYP2A6
SCHEMBL23287830 0.75 SNCA (0.43) MAPTSMN1; SMN2KDM4EMEN1ALDH1A1
SCHEMBL30080744 0.75 LIPG (0.55) LPLLIPGCYP2A6HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 56 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4685146-A1 COMPOUND FOR ORGANIC PHOTOVOLTAIC DEVICES, AND ORGANIC PHOTOVOLTAIC DEVICE, IMAGE SENSOR, AND ELECTRONIC DEVICE EACH CONTAINING SAME Duk San Neolux Co., Ltd. (KR) 2026-01-28 EP disclosed
EP-4536668-A1 PYRIDO[4,3-D]PYRIMIDINE DERIVATIVES AS KRAS INHIBITORS Bristol-Myers Squibb Company (US) 2025-04-16 EP disclosed
WO-2024225617-A1 COMPOUND FOR ORGANIC PHOTOVOLTAIC DEVICES, AND ORGANIC PHOTOVOLTAIC DEVICE, IMAGE SENSOR, AND ELECTRONIC DEVICE EACH CONTAINING SAME 덕산네오룩스 주식회사 2024-10-31 WO disclosed
US-20240334823-A1 ORGANOMETALLIC COMPOUND, ORGANIC LIGHT-EMITTING DEVICE INCLUDING ORGANOMETALLIC COMPOUND, AND ELECTRONIC APPARATUS INCLUDING ORGANIC LIGHT-EMITTING APPARATUS SAMSUNG DISPLAY CO., LTD. (KR) 2024-10-03 US disclosed
US-12052916-B2 Organometallic compound, organic light-emitting device including organometallic compound, and electronic apparatus including organic light-emitting apparatus SAMSUNG ELECTRONICS CO., LTD. (KR) 2024-07-30 US disclosed
US-20240067662-A1 KRAS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY 2024-02-29 US disclosed
US-20240067662-A1 KRAS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY 2024-02-29 US disclosed
US-20240067662-A1 KRAS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY 2024-02-29 US disclosed
WO-2023240188-A1 PYRIDO[4,3-D]PYRIMIDINE DERIVATIVES AS KRAS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2023-12-14 WO disclosed
WO-2023240188-A1 PYRIDO[4,3-D]PYRIMIDINE DERIVATIVES AS KRAS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2023-12-14 WO disclosed
US-20100298300-A1 TRIAZOLOPYRAZINE COMPOUNDS USEFUL FOR THE TREATMENT OF DEGENERATIVE & INFLAMMATORY DISEASES ANDREWS MARTIN JAMES INGLIS 2010-11-25 US disclosed
EP-2029602-B1 TRIAZOLOPYRAZINE COMPOUNDS USEFUL FOR THE TREATMENT OF DEGENERATIVE & INFLAMMATORY DISEASES GALAPAGOS NV (BE) 2010-04-21 EP disclosed
US-7501411-B2 Triazolopyrazine compounds useful for the treatment of degenerative and inflammatory diseases GALAPAGOS, NV (BE) 2009-03-10 US disclosed
EP-2029602-A2 TRIAZOLOPYRAZINE COMPOUNDS USEFUL FOR THE TREATMENT OF DEGENERATIVE & INFLAMMATORY DISEASES Galapagos N.V. (BE) 2009-03-04 EP disclosed
US-20090054454-A1 BENZOFURANYL- AND BENZOTHIENYL- PIPERAZINYL QUINOLINES AND METHODS OF THEIR USE VENKATESAN ARANAPAKAM MUDUMBAI 2009-02-26 US disclosed
US-20090054454-A1 BENZOFURANYL- AND BENZOTHIENYL- PIPERAZINYL QUINOLINES AND METHODS OF THEIR USE VENKATESAN ARANAPAKAM MUDUMBAI 2009-02-26 US disclosed
US-20080090818-A1 Triazolopyrazine compounds useful for the treatment of degenerative & inflammatory diseases GALAPAGOS NV (BE) 2008-04-17 US disclosed
WO-2007138072-A2 TRIAZOLOPYRAZINE COMPOUNDS USEFUL FOR THE TREATMENT OF DEGENERATIVE & INFLAMMATORY DISEASES GALAPAGOS N.V. (BE) 2007-12-06 WO disclosed
US-7276603-B2 serotonin receptor antagonists such as 8-{4-[2-(1-benzofuran-3-yl)ethyl]-1-piperazinyl}-6-fluoroquinoline, used for treatment and/or prevention of depression, anxiety and cognitive deficits arising from Alzheimer's disease, neurodegenerative disorders, schizophrenia and prostate cancer WYETH (US) 2007-10-02 US disclosed
US-7276603-B2 serotonin receptor antagonists such as 8-{4-[2-(1-benzofuran-3-yl)ethyl]-1-piperazinyl}-6-fluoroquinoline, used for treatment and/or prevention of depression, anxiety and cognitive deficits arising from Alzheimer's disease, neurodegenerative disorders, schizophrenia and prostate cancer WYETH (US) 2007-10-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100298300-A1 TRIAZOLOPYRAZINE COMPOUNDS USEFUL FOR THE TREATMENT OF DEGENERATIVE & INFLAMMATORY DISEASES P2RX5, P2RX3, IL1B MAPT 438/4885LPL 2158/4885LIPG 3151/4885
US-20240334823-A1 ORGANOMETALLIC COMPOUND, ORGANIC LIGHT-EMITTING DEVICE INCLUDING ORGANOMETALLIC COMPOUND, AND ELECTRONIC APPARATUS INCLUDING ORGANIC LIGHT-EMITTING APPARATUS L1CAM, MNS1, NOM1 MAPT 1313/4885LPL 1230/4885LIPG 2281/4885
US-20090054454-A1 BENZOFURANYL- AND BENZOTHIENYL- PIPERAZINYL QUINOLINES AND METHODS OF THEIR USE TPH1, TPH2, HTR2C MAPT 643/4885LPL 3217/4885LIPG 4522/4885
US-20240067662-A1 KRAS INHIBITORS KRAS, NRAS, HRAS MAPT 3872/4885LPL 3812/4885LIPG 2732/4885
US-12052916-B2 Organometallic compound, organic light-emitting device including organometallic compound, and electronic apparatus including organic light-emitting apparatus L1CAM, MNS1, NOM1 MAPT 1313/4885LPL 1230/4885LIPG 2281/4885
US-20080090818-A1 Triazolopyrazine compounds useful for the treatment of degenerative & inflammatory diseases P2RX5, P2RX3, IL1B MAPT 438/4885LPL 2158/4885LIPG 3151/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.