SCHEMBL574882

SCHEMBL574882

CN(CCO[Si](C)(C)C(C)(C)C)OCCc1ccc(F)cc1

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.41
AOC3 Q16853 1/20 0.40
ELOVL1 Q9BW60 2/20 0.39
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34
AQP1 P29972 1/20 0.34
SIGMAR1 Q99720 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1245973 0.84 ELOVL1 (0.41) TAAR1AOC3ELOVL1SIGMAR1
SCHEMBL9701242 0.72 HRH3 (0.42) TAAR1
SCHEMBL574561 0.72 TAAR1 (0.37) TAAR1ELOVL1SLC6A2SLC6A4SLC6A3
SCHEMBL19438939 0.71 SLC6A3 (0.43) TAAR1SLC6A2SLC6A4SLC6A3SIGMAR1
SCHEMBL1121430 0.71 IDO1 (0.50)
SCHEMBL2027168 0.70 LOXL2 (0.41)
SCHEMBL2696466 0.70 CYP1A2 (0.41) TAAR1
SCHEMBL503098 0.69 TAAR1 (0.33) TAAR1AOC3ELOVL1
SCHEMBL503485 0.69 TAAR1 (0.33) TAAR1AOC3ELOVL1
SCHEMBL574575 0.69 ADRB2 (0.35) ELOVL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2600853-A1 COMBINATIONS COMPRISING ATYPICAL ANTIPSYCHOTICS AND TAAR1 AGONISTS F.HOFFMANN-LA ROCHE AG (CH) 2013-06-12 EP disclosed
WO-2012016879-A1 COMBINATIONS COMPRISING ATYPICAL ANTIPSYCHOTICS AND TAAR1 AGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2012-02-09 WO disclosed