SCHEMBL5757754

SCHEMBL5757754

COc1ccc(Nc2nccc(N3CCCc4cccc(C)c43)n2)cc1OC

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTK2 Q05397 3/20 0.47
ALK Q9UM73 3/20 0.45
GSK3B P49841 2/20 0.45
CDK4 P11802 1/20 0.45
CDK2 P24941 1/20 0.45
BRD4 O60885 3/20 0.44
JAK2 O60674 3/20 0.43
AURKA O14965 3/20 0.43
FLT3 P36888 2/20 0.43
KIT P10721 1/20 0.43
IRAK4 Q9NWZ3 1/20 0.43
IGF1R P08069 2/20 0.43
PDGFRB P09619 2/20 0.42
AURKB Q96GD4 2/20 0.42
KDR P35968 2/20 0.42
DAPK3 O43293 1/20 0.42
PRKD3 O94806 1/20 0.42
MAP4K4 O95819 1/20 0.42
PAK4 O96013 1/20 0.42
ABL1 P00519 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5760237 0.90 PTK2 (0.58) PTK2ALKGSK3BJAK2AURKA
SCHEMBL5758741 0.87 L3MBTL1 (0.52) PTK2ALKCDK2AURKBKDR
SCHEMBL5759805 0.85 CDK2 (0.41) PTK2GSK3BCDK4CDK2KDR
SCHEMBL5761986 0.84 CDK4 (0.42) GSK3BCDK4CDK2BRD4JAK2
SCHEMBL5759742 0.84 SCN9A (0.42) PTK2GSK3BCDK4CDK2JAK2
SCHEMBL5760461 0.83 ROCK1 (0.40) PTK2CDK2JAK2AURKAKDR
SCHEMBL5757748 0.83 ALK (0.60) PTK2ALKGSK3BCDK4CDK2
SCHEMBL5758924 0.82 IDH1 (0.52) KDRFLT1ROCK1SYKL3MBTL1
SCHEMBL5760336 0.80 AURKA (0.45) JAK2AURKAAURKBJAK3SYK
SCHEMBL5760444 0.80 SYK (0.42) JAK2AURKAJAK3ROCK1SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242403-B1 2,4-DIAMINOPYRIMIDINE COMPOUNDS USFUL AS IMMUNOSUPPRESSANTS PFIZER PROD INC (US) 2006-01-04 EP claimed