SCHEMBL5758924

SCHEMBL5758924

Cc1cccc2c1N(c1ccnc(Nc3ccc(Oc4ccccc4)cc3)n1)CCC2

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 2/20 0.52
NR2C2 P49116 4/20 0.47
TAB1 Q15750 4/20 0.47
NFKB1 P19838 3/20 0.47
NFKB2 Q00653 3/20 0.47
RELA Q04206 3/20 0.47
PLK4 O00444 1/20 0.45
SCN9A Q15858 6/20 0.44
SCN5A Q14524 4/20 0.44
KCNH2 Q12809 3/20 0.44
KDR P35968 3/20 0.44
L3MBTL1 Q9Y468 1/20 0.41
FLT1 P17948 1/20 0.40
FLT4 P35916 1/20 0.40
IKBKB O14920 1/20 0.40
ROCK1 Q13464 1/20 0.39
SYK P43405 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5758741 0.90 L3MBTL1 (0.52) KDRL3MBTL1FLT1FLT4IKBKB
SCHEMBL5760461 0.86 ROCK1 (0.40) NR2C2TAB1NFKB1NFKB2RELA
SCHEMBL5758921 0.83 IDH1 (0.50) IDH1NR2C2TAB1NFKB1NFKB2
SCHEMBL5759805 0.82 CDK2 (0.41) KDRL3MBTL1FLT1FLT4SYK
SCHEMBL5757754 0.82 PTK2 (0.47) KDRL3MBTL1FLT1ROCK1SYK
SCHEMBL5761986 0.81 CDK4 (0.42) SCN9AKDR
SCHEMBL5759742 0.81 SCN9A (0.42) SCN9AKDRFLT1FLT4ROCK1
SCHEMBL5760237 0.80 PTK2 (0.58) KDRFLT1ROCK1SYK
SCHEMBL2373880 0.79 IDH1 (0.48) IDH1NR2C2TAB1NFKB1NFKB2
SCHEMBL5760262 0.78 CYP1A2 (0.45) PLK4KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242403-B1 2,4-DIAMINOPYRIMIDINE COMPOUNDS USFUL AS IMMUNOSUPPRESSANTS PFIZER PROD INC (US) 2006-01-04 EP claimed