SCHEMBL5758741

SCHEMBL5758741

COc1ccc(Nc2nccc(N3CCCc4cccc(C)c43)n2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.52
KDR P35968 5/20 0.50
CDK5 Q00535 3/20 0.47
CDK5R1 Q15078 2/20 0.47
PTK2 Q05397 3/20 0.46
MEN1 O00255 2/20 0.46
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
KMT2A Q03164 2/20 0.46
ALDH1A1 P00352 1/20 0.46
LMNA P02545 1/20 0.46
MAPT P10636 1/20 0.46
MAPK1 P28482 1/20 0.46
SYK P43405 1/20 0.44
LCK P06239 1/20 0.44
SRC P12931 1/20 0.44
MAPK14 Q16539 1/20 0.44
AKT1 P31749 1/20 0.43
PLK1 P53350 1/20 0.43
AURKB Q96GD4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5758924 0.90 IDH1 (0.52) L3MBTL1KDRSYKFLT1FLT4
SCHEMBL5760461 0.88 ROCK1 (0.40) L3MBTL1KDRCDK5CDK5R1PTK2
SCHEMBL5757754 0.87 PTK2 (0.47) L3MBTL1KDRCDK5PTK2SYK
SCHEMBL5759805 0.87 CDK2 (0.41) L3MBTL1KDRCDK5CDK5R1PTK2
SCHEMBL5760237 0.85 PTK2 (0.58) KDRCDK5PTK2SYKLCK
SCHEMBL5761986 0.83 CDK4 (0.42) KDRNPC1RAB9AAURKBPIK3CA
SCHEMBL5759742 0.83 SCN9A (0.42) KDRCDK5CDK5R1PTK2SYK
SCHEMBL5758463 0.81 KDR (0.55) KDRCDK5CDK5R1PTK2MEN1
SCHEMBL5760262 0.80 CYP1A2 (0.45) KDRSRCCDK2
SCHEMBL5760336 0.79 AURKA (0.45) MEN1KMT2AMAPTSYKAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242403-B1 2,4-DIAMINOPYRIMIDINE COMPOUNDS USFUL AS IMMUNOSUPPRESSANTS PFIZER PROD INC (US) 2006-01-04 EP claimed