SCHEMBL5760262

SCHEMBL5760262

Cc1cccc2c1N(c1ccnc(Nc3ccc(N4CCOCC4)nc3)n1)CCC2

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.45
SMG1 Q96Q15 3/20 0.44
CDK2 P24941 2/20 0.44
CDK1 P06493 1/20 0.44
JAK1 P23458 1/20 0.44
JAK3 P52333 1/20 0.44
ZAP70 P43403 1/20 0.43
PLK4 O00444 5/20 0.42
MTOR P42345 1/20 0.42
JAK2 O60674 4/20 0.41
FGFR1 P11362 1/20 0.41
KDR P35968 1/20 0.41
EPHB4 P54760 1/20 0.41
FGFR2 P21802 1/20 0.41
FGFR3 P22607 1/20 0.41
CCNK O75909 1/20 0.40
CCNA2 P20248 1/20 0.40
CCND3 P30281 1/20 0.40
CDK9 P50750 1/20 0.40
CDK6 Q00534 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5760255 0.84 SMG1 (0.44) CYP1A2SMG1CDK2CDK1JAK1
SCHEMBL5759805 0.83 CDK2 (0.41) CDK2CDK1MTORFGFR1KDR
SCHEMBL5760461 0.81 ROCK1 (0.40) CDK2JAK3PLK4JAK2KDR
SCHEMBL5758741 0.80 L3MBTL1 (0.52) CDK2KDRSRC
SCHEMBL5761986 0.79 CDK4 (0.42) CDK2JAK3JAK2KDR
SCHEMBL5759742 0.79 SCN9A (0.42) SMG1CDK2CDK1JAK3JAK2
SCHEMBL5759581 0.79 ROCK1 (0.55) ZAP70
SCHEMBL5758924 0.78 IDH1 (0.52) PLK4KDR
SCHEMBL5757754 0.77 PTK2 (0.47) CDK2JAK1JAK3JAK2FGFR1
SCHEMBL5760158 0.77 IGF1R (0.43) KDRPDGFRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242403-B1 2,4-DIAMINOPYRIMIDINE COMPOUNDS USFUL AS IMMUNOSUPPRESSANTS PFIZER PROD INC (US) 2006-01-04 EP claimed