SCHEMBL5775162

SCHEMBL5775162

O=C(O)CCc1c2c(nn1-c1ccccn1)CCCC2

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
FFAR4 Q5NUL3 14/20 0.45
KDM4E B2RXH2 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
HPGD P15428 1/20 0.43
RECQL P46063 1/20 0.43
HSD17B10 Q99714 1/20 0.43
NTRK1 P04629 1/20 0.41
GABRA1 P14867 1/20 0.40
GABRG2 P18507 1/20 0.40
GABRB3 P28472 1/20 0.40
GABRA3 P34903 1/20 0.40
ALDH1A1 P00352 1/20 0.39
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5774355 0.84 FABP4 (0.47) KDM4ENTRK1ALDH1A1
SCHEMBL5773019 0.76 RXRA (0.46) GABRA1
SCHEMBL4971846 0.75 GABRA1 (0.44) KDM4EHPGDHSD17B10NTRK1GABRA1
SCHEMBL29871089 0.75 GABRA1 (0.44) KDM4EHPGDHSD17B10NTRK1GABRA1
Hydrochloric Acid SCHEMBL30337257 0.74 GABRA1 (0.43) KDM4EHPGDHSD17B10NTRK1GABRA1
SCHEMBL15867016 0.72 GABRA1 (0.41) KDM4EHPGDHSD17B10NTRK1GABRA1
SCHEMBL5772957 0.71 POLB (0.55) KDM4EALDH1A1TDP1
SCHEMBL5777813 0.70 DRD2 (0.53) CYP3A4CYP2C9
SCHEMBL13974475 0.70 MAPT (0.46) KDM4EHPGDHSD17B10NTRK1GABRA1
SCHEMBL30337063 0.66 CD274 (0.40) HSD17B10GABRA1GABRG2GABRB3GABRA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0885883-B1 FUSED HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL APPLICATIONS THEREOF MITSUBISHI PHARMA CORP (JP) 2006-11-02 EP disclosed
US-6187774-B1 N-PIPERAZINYLALKYLINDAZOLE DERIVATIVES; PSYCHOLOGICAL DISORDERS, SCHIZOPHRENIA; SIDE EFFECT REDUCTION YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 2001-02-13 US disclosed
EP-0885883-A1 FUSED HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL APPLICATIONS THEREOF YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1998-12-23 EP disclosed