SCHEMBL5778129

SCHEMBL5778129

COC(=O)OB(OC(=O)OC)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.44
TSHR P16473 3/20 0.43
HSD17B10 Q99714 2/20 0.43
KDM4E B2RXH2 1/20 0.43
HPGD P15428 1/20 0.43
KCNN4 O15554 1/20 0.39
NAPRT Q6XQN6 1/20 0.39
CES2 O00748 1/20 0.38
CES1 P23141 1/20 0.38
ALDH1A1 P00352 1/20 0.37
GAA P10253 1/20 0.37
HTT P42858 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
HSD11B1 P28845 1/20 0.37
CYP3A4 P08684 1/20 0.36
ALOX5 P09917 1/20 0.36
SRC P12931 1/20 0.36
BCAT1 P54687 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1237453 0.82 KMT2A (0.42) KMT2ATSHRHSD17B10KDM4EHPGD
Hydrochloric Acid SCHEMBL3987325 0.80 KMT2A (0.41) KMT2ATSHRHSD17B10KDM4EHPGD
SCHEMBL6829989 0.79 TSHR (0.46) KMT2ATSHRHSD17B10ALDH1A1GAA
SCHEMBL9621660 0.78 ALDH1A1 (0.44) TSHRHSD17B10KDM4EHPGDNAPRT
SCHEMBL918997 0.78 ORAI1 (0.42) TSHRHSD17B10NAPRTCES2CES1
Biphenyl SCHEMBL28688628 0.78 MGLL (0.43) KMT2ATSHRHSD17B10KDM4EHPGD
SCHEMBL384013 0.74 ORAI1 (0.42) TSHRNAPRTCES2CES1ALDH1A1
SCHEMBL1712461 0.73 ELANE (0.46) TSHRHSD17B10KDM4EHPGDNAPRT
SCHEMBL3871760 0.73 KMT2A (0.47) KMT2AHSD17B10HPGDALDH1A1GAA
SCHEMBL28291707 0.72 MGLL (0.51) KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678138-A1 PYRIDINE COMPOUNDS AS INHIBITORS OF DIPEPTIDYL PEPTIDASE IV Takeda Pharmaceutical Company Limited (JP) 2006-07-12 EP disclosed
WO-2005042488-A1 PYRIDINE COMPOUNDS AS INHIBITORS OF DIPEPTIDYL PEPTIDASE IV TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2005-05-12 WO disclosed