SCHEMBL5808749

SCHEMBL5808749

CC(C)CN(Nc1ccnc(C#N)n1)C(=O)Cc1ccc(N(C)C)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1G O43497 4/20 0.37
CACNA1H O95180 4/20 0.37
CACNA1I Q9P0X4 4/20 0.37
ALDH1A1 P00352 3/20 0.34
KMT2A Q03164 1/20 0.34
CTSK P43235 2/20 0.34
CTSL P07711 1/20 0.34
CTSB P07858 1/20 0.34
CTSS P25774 1/20 0.34
HDAC1 Q13547 1/20 0.34
FGFR4 P22455 1/20 0.33
PANK3 Q9H999 1/20 0.33
PAK4 O96013 2/20 0.33
ACACB O00763 2/20 0.32
MMP3 P08254 1/20 0.32
MAPT P10636 2/20 0.31
KDM4E B2RXH2 1/20 0.31
TP53 P04637 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5792194 0.84 CXCR3 (0.37) CACNA1GCACNA1HCACNA1IKMT2APANK3
SCHEMBL5806357 0.78 FGFR4 (0.37) CTSKCTSLCTSBCTSSFGFR4
SCHEMBL5809045 0.77 CTSK (0.45) KMT2ACTSKCTSLCTSSFGFR4
SCHEMBL8270011 0.77 ALDH1A1 (0.39) CACNA1GCACNA1HCACNA1IALDH1A1KMT2A
SCHEMBL5793159 0.76 CTSK (0.36) CACNA1GCACNA1HCACNA1IALDH1A1KMT2A
Trifluoroacetic Acid SCHEMBL5791860 0.74 CTSS (0.36) CTSKCTSSPAK4
SCHEMBL5804565 0.73 CTSK (0.42) CTSKCTSLCTSBCTSSPANK3
Trifluoroacetic Acid SCHEMBL5808906 0.73 HRH4 (0.34) CTSKCTSSFGFR4PAK4
SCHEMBL8268861 0.69 CTSK (0.42) CTSKCTSLCTSBCTSSFGFR4
Trifluoroacetic Acid SCHEMBL5791245 0.68 CTSS (0.41) CTSKCTSLCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006027211-A1 2,4-SUBSTITUTED PYRIMIDINES AS CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2006-03-16 WO claimed