SCHEMBL5798138

SCHEMBL5798138

CCOC(=O)Cc1cccc(NS(=O)(=O)c2cccc(C)c2)n1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
KMT2A Q03164 7/20 0.52
MEN1 O00255 5/20 0.52
HSD11B1 P28845 1/20 0.49
HIF1A Q16665 1/20 0.45
PKM P14618 2/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC8 Q9BY41 1/20 0.45
HPGD P15428 2/20 0.44
MAPT P10636 1/20 0.44
POLB P06746 1/20 0.44
KDM4E B2RXH2 1/20 0.43
HSD17B10 Q99714 1/20 0.43
TDP1 Q9NUW8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5794528 0.88 PKM (0.53) ALDH1A1CYP2C9CYP2C19KMT2AMEN1
SCHEMBL5797968 0.87 KMT2A (0.68) ALDH1A1CYP2C9CYP2C19KMT2AMEN1
SCHEMBL5811010 0.81 KMT2A (0.61) ALDH1A1CYP2C9CYP2C19KMT2AMEN1
SCHEMBL5794952 0.80 HSD11B1 (0.53) ALDH1A1CYP2C9CYP2C19KMT2AMEN1
SCHEMBL5693072 0.78 HSD11B1 (0.76) ALDH1A1CYP2C9CYP2C19KMT2AMEN1
SCHEMBL5806893 0.78 CDK5 (0.49) ALDH1A1CYP2C9CYP2C19KMT2AMEN1
SCHEMBL30416934 0.77 CTPS1 (0.57) ALDH1A1CYP2C9CYP2C19KMT2AMEN1
SCHEMBL21381652 0.77 CTPS1 (0.57) ALDH1A1CYP2C9CYP2C19KMT2AMEN1
SCHEMBL5736794 0.76 LMNA (0.44) ALDH1A1CYP2C9CYP2C19KMT2AMEN1
SCHEMBL7044048 0.75 LMNA (0.43) ALDH1A1CYP2C9CYP2C19KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006050908-A1 INHIBITORS OF 11ΒΕΤΑ-HYDROXY STEROID DEHYDROGENASE TYPE 1 (11BETA-HSD1) EVOTEC AG (DE) 2006-05-18 WO disclosed