SCHEMBL579944

SCHEMBL579944

CCCCCNCCc1ccc(Oc2cc[c]cc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 0.55
S1PR2 O95136 3/20 0.45
S1PR1 P21453 3/20 0.45
S1PR3 Q99500 3/20 0.45
S1PR4 O95977 2/20 0.45
HRH3 Q9Y5N1 2/20 0.41
HRH4 Q9H3N8 1/20 0.41
LTA4H P09960 1/20 0.40
EPHX2 P34913 1/20 0.40
CHRM2 P08172 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C19 P33261 1/20 0.39
ADRB2 P07550 1/20 0.38
ADORA3 P0DMS8 1/20 0.38
CHRM1 P11229 1/20 0.38
ADRA2B P18089 1/20 0.38
ADRA2C P18825 1/20 0.38
DRD1 P21728 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9011773 0.83 ESR1 (0.50) CHRM2SMN1; SMN2ADORA3CHRM1ADRA2B
SCHEMBL921443 0.82 LTA4H (0.43) S1PR1S1PR3LTA4HCHRM2SMN1; SMN2
SCHEMBL919861 0.79 THRB (0.43) LTA4HALDH1A1LMNA
SCHEMBL16892534 0.78 SIGMAR1 (0.56) SIGMAR1S1PR2S1PR1S1PR3S1PR4
SCHEMBL16892525 0.78 SIGMAR1 (0.56) SIGMAR1S1PR2S1PR1S1PR3S1PR4
SCHEMBL580383 0.77 ADRB2 (0.51) SIGMAR1S1PR2S1PR1S1PR3S1PR4
SCHEMBL579438 0.76 ADRB2 (0.50) SIGMAR1S1PR2S1PR1S1PR3S1PR4
SCHEMBL16892602 0.74 SIGMAR1 (0.50) SIGMAR1S1PR2S1PR1S1PR3S1PR4
SCHEMBL5316000 0.73 KMT2A (0.53) S1PR2S1PR1S1PR3LTA4HDRD3
SCHEMBL475118 0.73 ALDH1A1 (0.57) LTA4HCHRM2SMN1; SMN2ADORA3CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1735268-B1 OPIOID RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2012-02-15 EP claimed