SCHEMBL5804565

SCHEMBL5804565

CC(C)CN(Nc1ccnc(C#N)n1)C(=O)N1CCN(C)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 6/20 0.42
CTSS P25774 3/20 0.42
CTSL P07711 2/20 0.42
CTSB P07858 1/20 0.42
HRH4 Q9H3N8 2/20 0.35
PAK4 O96013 2/20 0.35
KDM4E B2RXH2 1/20 0.35
ABL1 P00519 1/20 0.35
RIN1 Q13671 1/20 0.35
KDR P35968 2/20 0.34
GPR119 Q8TDV5 1/20 0.34
PANK3 Q9H999 2/20 0.33
ROCK2 O75116 2/20 0.33
ROCK1 Q13464 2/20 0.33
CDC42BPB Q9Y5S2 2/20 0.33
CDK8 P49336 2/20 0.33
CCNC P24863 1/20 0.33
MAP4K2 Q12851 1/20 0.33
HASPIN Q8TF76 1/20 0.33
CDK19 Q9BWU1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5806357 0.79 FGFR4 (0.37) CTSKCTSSCTSLCTSBPAK4
SCHEMBL5809045 0.76 CTSK (0.45) CTSKCTSSCTSLPAK4GPR119
SCHEMBL5791415 0.76 CTSK (0.47) CTSKCTSSCTSLCTSBHRH4
SCHEMBL5808749 0.73 CACNA1G (0.37) CTSKCTSSCTSLCTSBPAK4
SCHEMBL5792194 0.70 CXCR3 (0.37) PANK3
Trifluoroacetic Acid SCHEMBL5791860 0.68 CTSS (0.36) CTSKCTSSPAK4
SCHEMBL19116510 0.67 SMN1; SMN2 (0.57) CTSK
SCHEMBL8270031 0.67 CTSK (0.72) CTSKCTSSCTSLCTSBABL1
SCHEMBL5794243 0.65 CTSS (0.39) CTSKCTSSCTSLCTSB
SCHEMBL4137242 0.65 HRH4 (0.50) CTSKHRH4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006027211-A1 2,4-SUBSTITUTED PYRIMIDINES AS CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2006-03-16 WO disclosed