SCHEMBL5809045

SCHEMBL5809045

CC(C)CN(Nc1ccnc(C#N)n1)C(=O)CC1CCCC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 4/20 0.45
OPRM1 P35372 2/20 0.38
OPRL1 P41146 2/20 0.38
CTSS P25774 5/20 0.35
CTSL P07711 2/20 0.35
PAK4 O96013 2/20 0.33
MMP3 P08254 1/20 0.33
KMT2A Q03164 2/20 0.32
FGFR4 P22455 1/20 0.32
MAPK8 P45983 1/20 0.32
TSHR P16473 2/20 0.32
FFAR4 Q5NUL3 1/20 0.32
ADORA2A P29274 1/20 0.32
ADORA2B P29275 1/20 0.32
ADORA1 P30542 1/20 0.32
GPR119 Q8TDV5 1/20 0.32
MEN1 O00255 1/20 0.31
NPC1 O15118 1/20 0.31
TP53 P04637 1/20 0.31
RAB9A P51151 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5806357 0.78 FGFR4 (0.37) CTSKOPRM1OPRL1CTSSCTSL
SCHEMBL5808749 0.77 CACNA1G (0.37) CTSKCTSSCTSLPAK4MMP3
SCHEMBL5804565 0.76 CTSK (0.42) CTSKCTSSCTSLPAK4GPR119
SCHEMBL5792335 0.76 CTSK (0.37) CTSKOPRM1OPRL1CTSSCTSL
Trifluoroacetic Acid SCHEMBL5808906 0.74 HRH4 (0.34) CTSKOPRM1OPRL1CTSSPAK4
SCHEMBL5792194 0.73 CXCR3 (0.37) KMT2AMEN1SMN1; SMN2
Trifluoroacetic Acid SCHEMBL5791860 0.71 CTSS (0.36) CTSKCTSSPAK4MAPK8
SCHEMBL5791458 0.70 KMT2A (0.41) CTSKCTSSCTSLKMT2ATSHR
SCHEMBL8270526 0.70 CTSK (0.36) CTSKOPRM1OPRL1CTSSCTSL
SCHEMBL5794349 0.69 CTSK (0.39) CTSKCTSSCTSLFGFR4ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006027211-A1 2,4-SUBSTITUTED PYRIMIDINES AS CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2006-03-16 WO disclosed