SCHEMBL5828276

SCHEMBL5828276

O=C1c2ccc3[nH]c4ccccc4c3c2C(=O)N1CCO

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.51
CHEK1 O14757 2/20 0.47
HEXA P06865 1/20 0.44
HEXB P07686 1/20 0.44
NQO1 P15559 1/20 0.44
MAPT P10636 4/20 0.43
MEN1 O00255 3/20 0.43
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
KMT2A Q03164 3/20 0.43
AVPR1A P37288 1/20 0.43
ALDH1A1 P00352 4/20 0.43
PKM P14618 1/20 0.43
HSD17B10 Q99714 1/20 0.43
PRKCA P17252 2/20 0.43
KDM4E B2RXH2 2/20 0.42
HPGD P15428 1/20 0.40
RGS12 O14924 1/20 0.40
LMNA P02545 1/20 0.40
PABPC1 P11940 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9622936 0.84 TERT (0.52) PARP1HEXAHEXBNQO1MAPT
Hydrochloric Acid SCHEMBL9622732 0.83 TERT (0.51) PARP1HEXAHEXBNQO1MAPT
SCHEMBL8133497 0.83 SIRT1 (0.49) PARP1CHEK1HEXAHEXBNQO1
SCHEMBL9622806 0.82 NQO1 (0.67) PARP1CHEK1NQO1MAPTMEN1
SCHEMBL9622882 0.81 MEN1 (0.48) CHEK1MAPTMEN1NPC1RAB9A
SCHEMBL5828670 0.80 PARP1 (0.59) PARP1MAPTMEN1KMT2AALDH1A1
SCHEMBL7985172 0.80 SIRT1 (0.44) PARP1CHEK1HEXAHEXBNQO1
SCHEMBL6229657 0.79 PRKCA (0.63) PARP1CHEK1NQO1MAPTMEN1
SCHEMBL8560926 0.77 PARP1 (0.39) PARP1CHEK1NQO1MAPTMEN1
SCHEMBL8555782 0.77 PARP1 (0.41) PARP1CHEK1HEXAHEXBNQO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7094798-B1 Inhibitors of checkpoint kinases (Wee1 and Chk1) PFIZER INC (US) 2006-08-22 US claimed