SCHEMBL5828670

SCHEMBL5828670

CN1C(=O)c2ccc3[nH]c4ccccc4c3c2C1=O

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.59
ROCK2 O75116 1/20 0.47
ADORA3 P0DMS8 1/20 0.46
ADORA2A P29274 1/20 0.46
ADORA2B P29275 1/20 0.46
ADORA1 P30542 1/20 0.46
PRKCA P17252 3/20 0.45
SIRT2 Q8IXJ6 1/20 0.45
SIRT1 Q96EB6 1/20 0.45
GABRP O00591 1/20 0.44
GABRD O14764 1/20 0.44
GABRA1 P14867 1/20 0.44
GABRB1 P18505 1/20 0.44
GABRG2 P18507 1/20 0.44
GABRB3 P28472 1/20 0.44
GABRA5 P31644 1/20 0.44
GABRA3 P34903 1/20 0.44
GABRA2 P47869 1/20 0.44
GABRB2 P47870 1/20 0.44
GABRA4 P48169 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6229657 0.83 PRKCA (0.63) PARP1ROCK2PRKCAGABRPGABRD
SCHEMBL5828276 0.80 PARP1 (0.51) PARP1ROCK2PRKCAGABRPGABRD
SCHEMBL9622936 0.80 TERT (0.52) PARP1MEN1KMT2AKDM4EALDH1A1
Hydrochloric Acid SCHEMBL9622732 0.79 TERT (0.51) PARP1MEN1KMT2AKDM4EALDH1A1
SCHEMBL5438544 0.79 PRKCA (0.71) PARP1ROCK2ADORA3ADORA2AADORA2B
SCHEMBL25835901 0.78 PARP1 (0.68) PARP1PRKCAGABRPGABRDGABRA1
SCHEMBL25835900 0.78 PARP1 (0.68) PARP1PRKCAGABRPGABRDGABRA1
SCHEMBL9622806 0.77 NQO1 (0.67) PARP1ADORA3PRKCASIRT2MEN1
SCHEMBL8133497 0.76 SIRT1 (0.49) PARP1SIRT1MAPT
SCHEMBL14708732 0.76 ROCK2 (0.58) PARP1ROCK2ADORA3ADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7094798-B1 Inhibitors of checkpoint kinases (Wee1 and Chk1) PFIZER INC (US) 2006-08-22 US disclosed