SCHEMBL5828705

SCHEMBL5828705

COc1ccc(N(C)N(C)CC(O)c2ccc(O)c(O)c2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 2/20 0.50
CCNE2 O96020 1/20 0.42
CCNE1 P24864 1/20 0.42
CDK2 P24941 1/20 0.42
MAPT P10636 7/20 0.42
TDP1 Q9NUW8 6/20 0.42
ADRB2 P07550 6/20 0.42
KDM4E B2RXH2 5/20 0.42
ADRB1 P08588 5/20 0.42
MEN1 O00255 4/20 0.42
KMT2A Q03164 4/20 0.42
CYP3A4 P08684 4/20 0.42
ADRB3 P13945 4/20 0.42
MAPK1 P28482 4/20 0.42
TSHR P16473 4/20 0.42
RECQL P46063 3/20 0.42
APEX1 P27695 3/20 0.42
ADORA3 P0DMS8 3/20 0.42
DRD2 P14416 3/20 0.42
ADRA1D P25100 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5828703 0.76 AOC3 (0.50) AOC3CCNE2CCNE1CDK2MAPT
SCHEMBL521779 0.73 MAPT (0.58) MAPTTDP1ADRB2KDM4EADRB1
SCHEMBL521780 0.73 MAPT (0.58) MAPTTDP1ADRB2KDM4EADRB1
SCHEMBL17053665 0.72 MAPT (0.56) MAPTTDP1ADRB2KDM4EADRB1
SCHEMBL9768301 0.71 MAPT (0.68) AOC3MAPTTDP1ADRB2KDM4E
SCHEMBL5828700 0.71 ADRA1A (0.50) AOC3MAPTTDP1ADRB2KDM4E
SCHEMBL8690259 0.70 AKR1C3 (0.51) MAPTTDP1MEN1KMT2ATSHR
SCHEMBL11155392 0.70 ADRB2 (0.50) AOC3TDP1ADRB2ADRB1CYP3A4
SCHEMBL6479388 0.70 AOC3 (0.74) AOC3MAPTALDH1A1LMNAPOLB
SCHEMBL25100809 0.69 TDP1 (0.53) MAPTTDP1ADRB2KDM4EADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7109330-B2 Purine inhibitors of cyclin dependent kinase 2 and IκB-α CV THERAPEUTICS, INC. (US) 2006-09-19 US disclosed
US-20050080261-A1 Purine inhibitors of cyclin dependent kinase 2 and IkappaB-alpha LUM ROBERT T (US) 2005-04-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050080261-A1 Purine inhibitors of cyclin dependent kinase 2 and IkappaB-alpha IKBKB, NFKB1, CDK4 AOC3 3587/4885CCNE2 65/4885CCNE1 51/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.