SCHEMBL5833430

SCHEMBL5833430

COc1cc(N(CC2C3CCC2N(Cc2ccccc2)C3)C(=O)O)cc(OC)c1OC

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
ACHE P22303 5/20 0.41
BCHE P06276 3/20 0.41
BACE1 P56817 2/20 0.41
POLB P06746 1/20 0.40
CHRM2 P08172 1/20 0.39
CHRM3 P20309 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5833112 0.82 ROCK2 (0.41) ACHECHRM2CHRM3
SCHEMBL5833278 0.81 RNF4 (0.42) ACHECHRM2CHRM3
SCHEMBL5833539 0.81 CHRM2 (0.47) SIGMAR1CHRM2CHRM3
SCHEMBL5833452 0.80 DCUN1D1 (0.40) SIGMAR1MEN1KMT2AACHE
SCHEMBL5833435 0.80 SIGMAR1 (0.42) SIGMAR1MEN1KMT2AACHEBCHE
SCHEMBL5833937 0.80 OPRD1 (0.47) KMT2AACHECHRM2CHRM3
SCHEMBL4244062 0.78 SIGMAR1 (0.48) SIGMAR1ACHECHRM3
SCHEMBL5832943 0.77 ALPL (0.54) SIGMAR1MEN1KMT2AACHEBCHE
SCHEMBL5833269 0.77 KDM1A (0.40) MEN1KMT2A
SCHEMBL5833024 0.77 BRD4 (0.38) SIGMAR1MEN1KMT2ACHRM2CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7008955-B2 (2-azabicyclo[2.2.1]hept-7yl) methanol derivatives as nicotinic acetylcholine receptor agonists MERCK PATENT GMBH (DE) 2006-03-07 US claimed