SCHEMBL5833539

SCHEMBL5833539

O=C(O)N(CC1C2CCC1N(Cc1ccccc1)C2)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 2/20 0.47
CHRM3 P20309 2/20 0.47
OPRM1 P35372 5/20 0.43
OPRK1 P41145 5/20 0.43
BRD4 O60885 1/20 0.39
CCR5 P51681 1/20 0.38
MAPT P10636 1/20 0.38
SIGMAR1 Q99720 2/20 0.38
ROCK2 O75116 1/20 0.37
ARHGDIA P52565 1/20 0.37
ROCK1 Q13464 1/20 0.37
CHRM5 P08912 1/20 0.37
CHRM1 P11229 1/20 0.37
PKM P14618 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5833112 0.86 ROCK2 (0.41) CHRM2CHRM3OPRM1OPRK1BRD4
SCHEMBL5833024 0.85 BRD4 (0.38) CHRM2CHRM3OPRM1OPRK1BRD4
SCHEMBL5833937 0.84 OPRD1 (0.47) CHRM2CHRM3OPRM1OPRK1BRD4
SCHEMBL5833278 0.83 RNF4 (0.42) CHRM2CHRM3CHRM1
SCHEMBL5833269 0.83 KDM1A (0.40)
SCHEMBL5833452 0.82 DCUN1D1 (0.40) SIGMAR1
SCHEMBL5833430 0.81 SIGMAR1 (0.43) CHRM2CHRM3SIGMAR1
SCHEMBL5844904 0.81 LMNA (0.38) CHRM2CHRM3MAPTSIGMAR1ROCK2
SCHEMBL5833542 0.78 CHRM3 (0.44) CHRM2CHRM3OPRM1OPRK1BRD4
SCHEMBL5833003 0.77 SIGMAR1 (0.41) CHRM2CHRM3BRD4SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7008955-B2 (2-azabicyclo[2.2.1]hept-7yl) methanol derivatives as nicotinic acetylcholine receptor agonists MERCK PATENT GMBH (DE) 2006-03-07 US claimed