SCHEMBL5833112

SCHEMBL5833112

O=C(O)N(CC1C2CCC1N(Cc1ccccc1)C2)c1cc(Cl)nc(Cl)c1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.41
ARHGDIA P52565 1/20 0.41
ROCK1 Q13464 1/20 0.41
BRD4 O60885 1/20 0.36
ACHE P22303 3/20 0.36
PKM P14618 1/20 0.36
OPRD1 P41143 1/20 0.36
CHRM2 P08172 2/20 0.35
CHRM3 P20309 2/20 0.35
OPRM1 P35372 3/20 0.35
OPRK1 P41145 3/20 0.35
FAAH O00519 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5833539 0.86 CHRM2 (0.47) ROCK2ARHGDIAROCK1BRD4PKM
SCHEMBL5833278 0.84 RNF4 (0.42) ACHEOPRD1CHRM2CHRM3FAAH
SCHEMBL5833452 0.84 DCUN1D1 (0.40) ACHE
SCHEMBL5833430 0.82 SIGMAR1 (0.43) ACHECHRM2CHRM3
SCHEMBL5833024 0.82 BRD4 (0.38) ROCK2ARHGDIAROCK1BRD4PKM
SCHEMBL5833937 0.81 OPRD1 (0.47) BRD4ACHEOPRD1CHRM2CHRM3
SCHEMBL5833269 0.80 KDM1A (0.40) OPRD1FAAH
SCHEMBL5844904 0.78 LMNA (0.38) ROCK2ARHGDIAROCK1ACHECHRM2
SCHEMBL5833116 0.77 ROCK2 (0.41) ROCK2ARHGDIAROCK1BRD4PKM
SCHEMBL5833003 0.76 SIGMAR1 (0.41) BRD4ACHECHRM2CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7008955-B2 (2-azabicyclo[2.2.1]hept-7yl) methanol derivatives as nicotinic acetylcholine receptor agonists MERCK PATENT GMBH (DE) 2006-03-07 US claimed