SCHEMBL583885

SCHEMBL583885

N=C1OC(=N)c2c1ccc1c2OCO1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.38
TXNRD1 Q16881 1/20 0.34
TXNRD3 Q86VQ6 1/20 0.34
TXNRD2 Q9NNW7 1/20 0.34
DRD2 P14416 1/20 0.33
DRD1 P21728 1/20 0.33
AOC3 Q16853 2/20 0.33
ABCG2 Q9UNQ0 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HSD17B10 Q99714 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
NQO2 P16083 3/20 0.31
CYP19A1 P11511 2/20 0.31
CYP1A2 P05177 1/20 0.31
CYP1B1 Q16678 1/20 0.31
CYP3A4 P08684 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9488966 0.70 ALOX5 (0.47) PTGS2TXNRD1TXNRD3TXNRD2DRD2
SCHEMBL584571 0.69 CYP3A4 (0.38) PTGS2ABCG2ALDH1A1HSD17B10TDP1
SCHEMBL14302835 0.68 CYP1A2 (0.51) PTGS2DRD2DRD1ABCG2CYP1A2
SCHEMBL4596292 0.67 ABCG2 (0.40) PTGS2TXNRD1TXNRD3TXNRD2DRD2
SCHEMBL14179075 0.67 PTGS2 (0.40) PTGS2TXNRD1TXNRD3TXNRD2AOC3
SCHEMBL9206878 0.66 PARP1 (0.42) PTGS2TXNRD1TXNRD3TXNRD2AOC3
SCHEMBL1768496 0.64 PKM (0.39) PTGS2TXNRD1TXNRD3TXNRD2DRD2
SCHEMBL4596267 0.62 NQO2 (0.36) PTGS2TXNRD1TXNRD3TXNRD2DRD2
SCHEMBL23635064 0.62 TXNRD1 (0.40) PTGS2TXNRD1TXNRD3TXNRD2DRD2
SCHEMBL9348922 0.62 HSP90AA1 (0.39) TXNRD1TXNRD3TXNRD2DRD2DRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120077989-A1 CYCLIC IMIDATE LIGANDS UNIVERSITEIT GENT (BE) 2012-03-29 US disclosed
EP-2416879-A1 CYCLIC IMIDATE LIGANDS Universiteit Gent (BE) 2012-02-15 EP disclosed
WO-2010115903-A1 CYCLIC IMIDATE LIGANDS UNIVERSITEIT GENT (BE) 2010-10-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120077989-A1 CYCLIC IMIDATE LIGANDS IDH2, CYCS, NAPRT PTGS2 2952/4885TXNRD1 4473/4885TXNRD3 4131/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.