SCHEMBL5886950

SCHEMBL5886950

Cc1nc(N2CCc3ccccc3C2)nc2c1ccc(=O)n2-c1ccc(C(=O)NCC2CCCO2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 5/20 0.51
RAB9A P51151 3/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
LMNA P02545 2/20 0.51
POLB P06746 1/20 0.51
MAPT P10636 1/20 0.51
NAMPT P43490 4/20 0.47
ATM Q13315 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
ALDH1A1 P00352 5/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
KDM4E B2RXH2 4/20 0.42
CYP2C9 P11712 2/20 0.42
HTT P42858 2/20 0.42
HSD17B10 Q99714 2/20 0.42
CYP1A2 P05177 1/20 0.42
GLA P06280 1/20 0.42
CYP3A4 P08684 1/20 0.42
GAA P10253 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5886952 0.89 HPGD (0.58) HPGDRAB9ASMN1; SMN2LMNAPOLB
SCHEMBL5886901 0.88 NAPEPLD (0.45) POLBNAMPTMEN1KMT2AGAA
SCHEMBL5886978 0.87 HPGD (0.54) HPGDRAB9ASMN1; SMN2LMNAPOLB
SCHEMBL5887047 0.86 HPGD (0.54) HPGDRAB9ASMN1; SMN2LMNAPOLB
SCHEMBL5886750 0.83 ADAMTS4 (0.45) SMN1; SMN2LMNAPOLBMAPTNAMPT
SCHEMBL5887343 0.83 PRMT5 (0.43) RAB9ALMNAMAPTALDH1A1MEN1
SCHEMBL5887057 0.83 DRD2 (0.41) RAB9ASMN1; SMN2LMNAMAPTNPC1
SCHEMBL5886716 0.83 SMN1; SMN2 (0.41) HPGDRAB9ASMN1; SMN2LMNAPOLB
SCHEMBL5887620 0.82 HPGD (0.54) HPGDRAB9ASMN1; SMN2LMNAPOLB
SCHEMBL5887024 0.82 MAPT (0.44) HPGDRAB9ASMN1; SMN2LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7019002-B2 Substituted on 8th position with benzoic acid, ester or amide groups; anticancer agents PHARMACIA & UPJOHN, S.P.A. (IT) 2006-03-28 US claimed
US-20040009993-A1 Pyridopyrimidinones derivatives as telomerase inhibitors PHARMACIA ITALIA S.P.A. 2004-01-15 US claimed
US-7019002-B2 Substituted on 8th position with benzoic acid, ester or amide groups; anticancer agents PHARMACIA & UPJOHN, S.P.A. (IT) 2006-03-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040009993-A1 Pyridopyrimidinones derivatives as telomerase inhibitors TERT, TERF2, TERF2IP HPGD 1371/4885RAB9A 3217/4885SMN1; SMN2 2219/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.