SCHEMBL6004207

SCHEMBL6004207

CCc1ccc(Oc2ccnc3ccc(OCCO)cc23)c(-c2ccccn2)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP19A1 P11511 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
SLC22A12 Q96S37 1/20 0.36
ACSS2 Q9NR19 1/20 0.36
CBFB Q13951 1/20 0.36
KDM4E B2RXH2 1/20 0.35
NPC1 O15118 1/20 0.35
ALDH1A1 P00352 1/20 0.35
GLA P06280 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
PKM P14618 1/20 0.35
HPGD P15428 1/20 0.35
MAPK1 P28482 1/20 0.35
RAB9A P51151 1/20 0.35
ATM Q13315 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6004067 0.89 SLC22A12 (0.38) SLC22A12ACSS2PDE4APDE4DMET
SCHEMBL6005265 0.89 TGFBR1 (0.44) CYP1A2CYP2D6CYP19A1CYP2C9CYP2C19
SCHEMBL6004984 0.88 PDE3B (0.39) CBFBKDM4ENPC1ALDH1A1GLA
SCHEMBL6004710 0.87 CYP3A4 (0.42) CYP1A2CYP2C9ACSS2CBFBKDM4E
SCHEMBL6004800 0.85 KDR (0.40) ACSS2KDM4ENPC1ALDH1A1GLA
SCHEMBL6004082 0.85 CBFB (0.37) CBFBKDM4ENPC1ALDH1A1GAA
SCHEMBL6005438 0.84 MET (0.35) CBFBKDM4ENPC1ALDH1A1MAPT
SCHEMBL6002895 0.84 TGFBR1 (0.48) CYP1A2CYP2D6CYP19A1CYP2C9CYP2C19
SCHEMBL6004857 0.80 SRC (0.37) KDM4EALDH1A1GAAMAPTHPGD
SCHEMBL6002914 0.80 PDGFRB (0.49) METKDRMST1RTGFBR1EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1724268-A1 COMPOUND HAVING TGF-BETA INHIBITORY ACTIVITY AND PHARMACEUTICAL COMPOSITION CONTAINING SAME KIRIN BEER KABUSHIKI KAISHA (JP) 2006-11-22 EP disclosed