SCHEMBL6005265

SCHEMBL6005265

Cc1ccc(Oc2ccnc3ccc(OCCO)cc23)c(-c2ccccn2)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 4/20 0.44
SYK P43405 2/20 0.38
SLC22A12 Q96S37 1/20 0.37
PDE2A O00408 3/20 0.37
PDE10A Q9Y233 3/20 0.37
AURKB Q96GD4 1/20 0.36
INCENP Q9NQS7 1/20 0.36
KDM4E B2RXH2 1/20 0.36
NPC1 O15118 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP19A1 P11511 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
ACSS2 Q9NR19 1/20 0.35
MAOA P21397 1/20 0.35
CBFB Q13951 1/20 0.35
SRC P12931 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6004922 0.89 SLC22A12 (0.39) TGFBR1SYKSLC22A12PDE2APDE10A
SCHEMBL6004207 0.89 CYP1A2 (0.37) TGFBR1SLC22A12KDM4ENPC1CYP1A2
SCHEMBL6002895 0.87 TGFBR1 (0.48) TGFBR1SLC22A12PDE2APDE10AKDM4E
SCHEMBL6004827 0.86 CYP3A4 (0.44) TGFBR1SYKAURKBINCENPKDM4E
SCHEMBL6005251 0.84 PDE2A (0.39) TGFBR1SLC22A12PDE2APDE10AAURKB
SCHEMBL6005330 0.83 TGFBR1 (0.46) TGFBR1SYKAURKBINCENPKDM4E
SCHEMBL6005388 0.80 TGFBR1 (0.48) TGFBR1KDM4ENPC1MAOA
SCHEMBL6004162 0.79 ALDH1A1 (0.36) TGFBR1SYKAURKBINCENPSRC
SCHEMBL6004262 0.79 ALDH1A1 (0.36) TGFBR1SYKAURKBINCENPKDM4E
SCHEMBL6004343 0.79 SIGMAR1 (0.36) PDE2APDE10AMAOAEGFRBTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1724268-A1 COMPOUND HAVING TGF-BETA INHIBITORY ACTIVITY AND PHARMACEUTICAL COMPOSITION CONTAINING SAME KIRIN BEER KABUSHIKI KAISHA (JP) 2006-11-22 EP disclosed