SCHEMBL6004795

SCHEMBL6004795

Fc1cc2nccc(Oc3cc4cccnc4nc3-c3ccccc3)c2cc1F

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
FGFR2 P21802 2/20 0.36
MET P08581 5/20 0.36
KDR P35968 1/20 0.36
MST1R Q04912 1/20 0.36
MAPK14 Q16539 1/20 0.36
AXL P30530 1/20 0.36
TOP1 P11387 1/20 0.36
SRC P12931 1/20 0.34
TGFBR1 P36897 1/20 0.34
NPC1 O15118 1/20 0.34
DHODH Q02127 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6004093 0.91 MET (0.45) FGFR2METKDRMST1RAXL
SCHEMBL6004849 0.91 MET (0.45) FGFR2METKDRMST1RAXL
SCHEMBL6005302 0.88 DHODH (0.39) FGFR2MAPK14TOP1DHODH
SCHEMBL6004803 0.86 FGFR2 (0.36) FGFR2KDRAXLSRCTGFBR1
SCHEMBL6004276 0.86 LMNA (0.39) KDRTOP1NPC1DHODH
SCHEMBL3895779 0.85 FGFR2 (0.53) FGFR2KDRAXLSRCTGFBR1
SCHEMBL6005306 0.84 MAPK14 (0.34) METMST1RMAPK14TOP1NPC1
SCHEMBL6005353 0.83 CCNC (0.40) METKDRMAPK14TOP1DHODH
SCHEMBL6004765 0.83 FGFR2 (0.45) FGFR2KDRAXLSRCTGFBR1
SCHEMBL6004812 0.82 FGFR2 (0.44) FGFR2METKDRAXLSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1724268-A1 COMPOUND HAVING TGF-BETA INHIBITORY ACTIVITY AND PHARMACEUTICAL COMPOSITION CONTAINING SAME KIRIN BEER KABUSHIKI KAISHA (JP) 2006-11-22 EP disclosed