Clausine C

Clausine C

SCHEMBL601713

COC(=O)c1ccc2[nH]c3cc(OC)ccc3c2c1

nearest known ligand 0.67

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 3/20 0.67
MEN1 O00255 5/20 0.58
KMT2A Q03164 5/20 0.58
ALDH1A1 P00352 6/20 0.57
KDM4E B2RXH2 5/20 0.57
HSD17B10 Q99714 4/20 0.57
MAPT P10636 4/20 0.57
HPGD P15428 3/20 0.57
USP2 O75604 1/20 0.57
GAA P10253 1/20 0.57
ALOX15 P16050 1/20 0.57
NPSR1 Q6W5P4 1/20 0.57
TSHR P16473 1/20 0.56
GFER P55789 1/20 0.56
PARP1 P09874 2/20 0.53
MTNR1A P48039 1/20 0.53
MTNR1B P49286 1/20 0.53
RAB9A P51151 2/20 0.52
NPC1 O15118 1/20 0.52
CA1 P00915 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19331068 0.93 KDM4E (0.66) KIF11MEN1KMT2AALDH1A1KDM4E
SCHEMBL29373898 0.93 KDM4E (0.66) KIF11MEN1KMT2AALDH1A1KDM4E
SCHEMBL17461848 0.87 KIF11 (0.67) KIF11MEN1KMT2AALDH1A1KDM4E
SCHEMBL28063129 0.86 KIF11 (0.70) KIF11MEN1KMT2AALDH1A1KDM4E
SCHEMBL4725998 0.83 KIF11 (0.84) KIF11MEN1KMT2AALDH1A1KDM4E
SCHEMBL29708168 0.83 KIF11 (0.84) KIF11MEN1KMT2AALDH1A1KDM4E
SCHEMBL71508 0.82 KIF11 (0.82) KIF11MEN1KMT2AALDH1A1KDM4E
SCHEMBL600063 0.81 KIF11 (0.64) KIF11MEN1KMT2AALDH1A1KDM4E
SCHEMBL5795304 0.80 ABCG2 (0.53) KIF11MEN1KMT2AALDH1A1KDM4E
SCHEMBL6981871 0.79 ALDH1A1 (0.68) KIF11MEN1KMT2AALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3229811-B1 PREVENTION AND TREATMENT OF INFLAMMATORY CONDITIONS GRI BIO INC (US) 2021-02-24 EP disclosed
US-20170096426-A1 Novel Tricyclic Modulators of Cannabinoid Receptors THE UNIV OF MONTANA (US) 2017-04-06 US disclosed
US-20170096426-A1 Novel Tricyclic Modulators of Cannabinoid Receptors THE UNIV OF MONTANA (US) 2017-04-06 US disclosed
US-20170096426-A1 Novel Tricyclic Modulators of Cannabinoid Receptors THE UNIV OF MONTANA (US) 2017-04-06 US disclosed
WO-2016094226-A1 PREVENTION AND TREATMENT OF INFLAMMATORY CONDITIONS GLYCOREGIMMUNE, INC. (US) 2016-06-16 WO disclosed
US-20160158258-A1 PREVENTION AND TREATMENT OF INFLAMMATORY CONDITIONS ALTIUM GROWTH FUND, LP 2016-06-09 US disclosed
US-20120039804-A1 Novel Tricyclic Modulators of Cannabinoid Receptors NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2012-02-16 US disclosed
US-20120039804-A1 Novel Tricyclic Modulators of Cannabinoid Receptors NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2012-02-16 US disclosed
US-20120039804-A1 Novel Tricyclic Modulators of Cannabinoid Receptors NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2012-02-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120039804-A1 Novel Tricyclic Modulators of Cannabinoid Receptors CNR1, CNR2, OPRL1 KIF11 4554/4885MEN1 3607/4885KMT2A 1530/4885
US-20170096426-A1 Novel Tricyclic Modulators of Cannabinoid Receptors CNR1, CNR2, OPRL1 KIF11 4554/4885MEN1 3607/4885KMT2A 1530/4885
US-20160158258-A1 PREVENTION AND TREATMENT OF INFLAMMATORY CONDITIONS RXRA, RXRG, CX3CR1 KIF11 3113/4885MEN1 4785/4885KMT2A 411/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.