SCHEMBL6030680

SCHEMBL6030680

FC(F)(F)c1ccc2c(c1)N=Cc1c(cccc1N1CCNCC1)N2

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 2/20 0.46
HTR1D P28221 2/20 0.46
HTR2C P28335 2/20 0.46
HTR3E A5X5Y0 1/20 0.46
HTR3B O95264 1/20 0.46
ALDH1A1 P00352 1/20 0.46
HTR3D Q70Z44 1/20 0.46
HTR3C Q8WXA8 1/20 0.46
SIGMAR1 Q99720 1/20 0.46
MAPT P10636 1/20 0.45
THRB P10828 1/20 0.45
ADRB2 P07550 2/20 0.45
NCF1 P14598 2/20 0.45
HTR1A P08908 1/20 0.45
ADRB1 P08588 2/20 0.41
IDH2 P48735 1/20 0.40
CYP1A2 P05177 1/20 0.38
CHRM2 P08172 1/20 0.38
CHRM4 P08173 1/20 0.38
CYP3A4 P08684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5936567 0.86 HTR1A (0.44) HTR3AHTR1DHTR2CHTR1ACYP1A2
SCHEMBL5560257 0.84 ADRB2 (0.43) HTR3AHTR1DHTR2CHTR3EHTR3B
SCHEMBL5936594 0.84 NCF1 (0.41) HTR3AHTR1DHTR2CHTR3EHTR3B
SCHEMBL5936593 0.84 HTR1A (0.46) HTR3AHTR2CADRB2HTR1AADRB1
SCHEMBL4202572 0.84 CYP1A2 (0.55) HTR3AHTR1DHTR2CHTR3EHTR3B
SCHEMBL6029951 0.83 HTR1A (0.44) HTR3AHTR1DHTR2CHTR3EHTR3B
SCHEMBL6030820 0.83 DRD2 (0.45) HTR3AHTR1DHTR2CHTR3EHTR3B
SCHEMBL4331521 0.83 HTR3A (0.40) HTR3AHTR1DHTR2CHTR3EHTR3B
SCHEMBL5936575 0.82 HTR1A (0.47) HTR3AHTR1DHTR2CNCF1HTR1A
SCHEMBL4428815 0.81 ADRB1 (0.41) HTR3AHTR1DHTR2CHTR3EHTR3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1696931-A2 AMINO SUBSTITUTED DIARYL [A,D]CYCLOHEPTENE ANALOGS AS MUSCARINIC AGONISTS AND METHODS OF TREATMENT OF NEUROPSYCHIATRIC DISORDERS Acadia Pharmaceuticals Inc. (US) 2006-09-06 EP disclosed
WO-2005063254-A2 AMINO SUBSTITUTED DIARYL[A,D]CYCLOHEPTENE ANALOGS AS MUSCARINIC AGONISTS AND METHODS OF TREATMENT OF NEUROPSYCHIATRIC DISORDERS ACADIA PHARMACEUTICALS INC. (US) 2005-07-14 WO disclosed