SCHEMBL6077778

SCHEMBL6077778

CN1C(=O)C2CSC(=O)N2C(=O)C1c1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.37
TSHR P16473 1/20 0.37
BRD4 O60885 3/20 0.34
ALDH1A1 P00352 2/20 0.34
ATM Q13315 1/20 0.34
MMP2 P08253 1/20 0.33
LMNA P02545 3/20 0.33
PRCP P42785 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
SRD5A1 P18405 1/20 0.33
CHRNB2 P17787 1/20 0.33
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
CHRNA7 P36544 1/20 0.33
CHRNA4 P43681 1/20 0.33
MITF O75030 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
MAPT P10636 1/20 0.32
HTT P42858 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6078380 0.77 TACR1 (0.47) MAPT
SCHEMBL10540887 0.76 TSHR (0.47) KMT2ATSHRBRD4ALDH1A1MMP2
SCHEMBL27705342 0.75 ALDH1A1 (0.44) KMT2ATSHRBRD4ALDH1A1ATM
SCHEMBL6078979 0.74
SCHEMBL6079130 0.71
SCHEMBL6076752 0.71 LMNA (0.43) KMT2AALDH1A1LMNAADORA3MITF
SCHEMBL27686342 0.70 ALDH1A1 (0.40) KMT2AALDH1A1LMNAMITFTDP1
SCHEMBL6078230 0.70
SCHEMBL15125072 0.70 CHRNB2 (0.50) KMT2ATSHRALDH1A1LMNACHRNB2
SCHEMBL6077343 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7022317-B2 Heterocyclic derivatives of 2-oxothiazolidine-4-carboxylic acid, and use as active photoprotective agents L'OREAL (FR) 2006-04-04 US claimed
US-20050129635-A1 Novel heterocyclic derivatives of 2-oxothiazolidine-4-carboxylic acid, and use as active photoprotective agents L'OREAL S.A. (FR) 2005-06-16 US claimed
US-7022317-B2 Heterocyclic derivatives of 2-oxothiazolidine-4-carboxylic acid, and use as active photoprotective agents L'OREAL (FR) 2006-04-04 US disclosed
US-20050129635-A1 Novel heterocyclic derivatives of 2-oxothiazolidine-4-carboxylic acid, and use as active photoprotective agents L'OREAL S.A. (FR) 2005-06-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050129635-A1 Novel heterocyclic derivatives of 2-oxothiazolidine-4-carboxylic acid, and use as active photoprotective agents CUTA, OGDH, TYR KMT2A 2556/4885TSHR 4123/4885BRD4 1705/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.