SCHEMBL608552

SCHEMBL608552

O=[N+]([O-])c1ccc(O)c2c1OCO2

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TXNRD1 Q16881 1/20 0.53
TXNRD3 Q86VQ6 1/20 0.53
TXNRD2 Q9NNW7 1/20 0.53
SMN1; SMN2 Q16637 3/20 0.46
TP53 P04637 2/20 0.46
HPGD P15428 2/20 0.46
TSHR P16473 2/20 0.46
CTSB P07858 2/20 0.46
CYP3A4 P08684 1/20 0.46
HIF1A Q16665 1/20 0.46
GPR35 Q9HC97 4/20 0.43
MAPK1 P28482 2/20 0.43
ALDH1A1 P00352 2/20 0.43
L3MBTL1 Q9Y468 2/20 0.42
ALOX15 P16050 1/20 0.42
HSD17B10 Q99714 1/20 0.42
CDK2 P24941 2/20 0.40
MAPT P10636 5/20 0.40
POLB P06746 2/20 0.40
CASP6 P55212 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4491664 0.79 TXNRD1 (0.50) TXNRD1TXNRD3TXNRD2SMN1; SMN2HPGD
SCHEMBL29661290 0.78 TXNRD1 (0.53) TXNRD1TXNRD3TXNRD2SMN1; SMN2TSHR
SCHEMBL24327364 0.78 TXNRD1 (0.53) TXNRD1TXNRD3TXNRD2SMN1; SMN2TSHR
SCHEMBL5723712 0.78 TXNRD1 (0.53) TXNRD1TXNRD3TXNRD2TSHRCYP3A4
SCHEMBL28958003 0.78 TXNRD1 (0.53) TXNRD1TXNRD3TXNRD2SMN1; SMN2TP53
SCHEMBL3540216 0.77 TXNRD1 (0.49) TXNRD1TXNRD3TXNRD2SMN1; SMN2TSHR
SCHEMBL2265157 0.77 AOC3 (0.44) SMN1; SMN2HPGDCYP3A4HIF1AALDH1A1
SCHEMBL11032479 0.75 TXNRD1 (0.68) TXNRD1TXNRD3TXNRD2GPR35ALDH1A1
SCHEMBL4495775 0.75 TXNRD1 (0.54) TXNRD1TXNRD3TXNRD2SMN1; SMN2CYP3A4
SCHEMBL30077309 0.74 GPR35 (0.43) TXNRD1TXNRD3TXNRD2SMN1; SMN2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130157986-A1 NOVEL METHYLENEDIOXY PHENOLIC COMPOUNDS AND THEIR USE TO TREAT DISEASE INVASC THERAPEUTICS, INC. (US) 2013-06-20 US disclosed
EP-2539317-A2 DIHYDROLIPOIC ACID DERIVATIVES COMPRISING NITRIC OXIDE AND THERAPEUTIC USES THEREOF Invasc Therapeutics, Inc. (US) 2013-01-02 EP disclosed
US-8198317-B2 Methylenedioxy phenolic compounds and their use to treat disease THE OHIO STATE UNIVERSITY RESEARCH FOUNDATION (US) 2012-06-12 US disclosed
US-20120041025-A1 Dihydrolipoic Acid Derivatives Comprising Nitric Oxide and Therapeutic Uses Thereof CARMEL BIOSCIENCES, INC. 2012-02-16 US disclosed
EP-2324005-A1 NOVEL METHYLENEDIOXY PHENOLIC COMPOUNDS AND THEIR USE TO TREAT DISEASE The Ohio State University Research Foundation (US) 2011-05-25 EP disclosed
WO-2010096677-A2 DIHYDROLIPOIC ACID DERIVATIVES COMPRISING NITRIC OXIDE AND THERAPEUTIC USES THEREOF INVASC THERAPEUTICS, INC. (US) 2010-08-26 WO disclosed
WO-2010017323-A1 NOVEL METHYLENEDIOXY PHENOLIC COMPOUNDS AND THEIR USE TO TREAT DISEASE THE OHIO STATE UNIVERSITY RESEARCH FOUNDATION (US) 2010-02-11 WO disclosed
US-20100035849-A1 NOVEL METHYLENEDIOXY PHENOLIC COMPOUNDS AND THEIR USE TO TREAT DISEASE OHIO STATE UNIVERSITY RESEARCH FOUNDATION (US) 2010-02-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100035849-A1 NOVEL METHYLENEDIOXY PHENOLIC COMPOUNDS AND THEIR USE TO TREAT DISEASE REN, PCSK9, ALOX12 TXNRD1 1455/4885TXNRD3 663/4885TXNRD2 104/4885
US-20120041025-A1 Dihydrolipoic Acid Derivatives Comprising Nitric Oxide and Therapeutic Uses Thereof DLD, LDLR, ALOX15 TXNRD1 394/4885TXNRD3 355/4885TXNRD2 127/4885
US-20130157986-A1 NOVEL METHYLENEDIOXY PHENOLIC COMPOUNDS AND THEIR USE TO TREAT DISEASE REN, PCSK9, COMT TXNRD1 1560/4885TXNRD3 710/4885TXNRD2 121/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.