SCHEMBL6139412

SCHEMBL6139412

COCCc1cc[nH]c1C=O

nearest known ligand 0.32

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 1/20 0.32
TSHR P16473 1/20 0.30
CYP2A6 P11509 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8207936 1.00 ADRA1A (0.32) ADRA1ATSHRCYP2A6
SCHEMBL9225445 0.79 GPR84 (0.33)
SCHEMBL4053225 0.78
SCHEMBL7086196 0.75 GPR84 (0.45) TSHR
SCHEMBL8194399 0.71 HCAR2 (0.32)
SCHEMBL7482610 0.71 CA2 (0.32)
SCHEMBL4267778 0.71
SCHEMBL15794861 0.69 DAO (0.39) ADRA1ATSHR
SCHEMBL14560346 0.68 SRC (0.43) TSHR
SCHEMBL4171179 0.68 GABRA1 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1476423-A4 ARYLSULFONAMIDOBENZYLIC COMPOUNDS TULARIK INC (US) 2005-12-14 EP disclosed
EP-1476423-A2 ARYLSULFONAMIDOBENZYLIC COMPOUNDS Tularik Inc. (US) 2004-11-17 EP disclosed
WO-2003063576-A2 ARYLSULFONAMIDOBENZYLIC COMPOUNDS TULARIK INC. (US) 2003-08-07 WO disclosed