SCHEMBL6156220

SCHEMBL6156220

CO[C@@H]1[C@H](O)[C@@H](O)[C@H](c2ccc3c(N4CCNCC4)cc(=O)oc3c2C)O[C@]1(C)CO

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 2/20 0.46
PDE3A Q14432 2/20 0.46
PRKDC P78527 3/20 0.38
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA4 P22748 1/20 0.33
MAOB P27338 1/20 0.33
CA5A P35218 1/20 0.33
CA7 P43166 1/20 0.33
CA5B Q9Y2D0 1/20 0.33
CCNT1 O60563 1/20 0.33
CCNA2 P20248 1/20 0.33
CDK2 P24941 1/20 0.33
CDK9 P50750 1/20 0.33
BACE1 P56817 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6156060 0.90 PDE3B (0.37) PDE3BPDE3APRKDC
SCHEMBL6158814 0.89 PRKDC (0.37) PDE3BPDE3APRKDC
SCHEMBL6156871 0.89 KDM4E (0.42) PDE3BPDE3APRKDC
SCHEMBL8371288 0.88 PDE3B (0.39) PDE3BPDE3APRKDC
SCHEMBL6156255 0.87 MEN1 (0.38) PDE3BPDE3APRKDC
SCHEMBL6155515 0.86 RAB9A (0.33) PDE3BPDE3APRKDC
SCHEMBL6165736 0.86 PTPN1 (0.38) PDE3BPDE3APRKDC
SCHEMBL6156254 0.81 KDM4E (0.35) CA12MAOB
SCHEMBL6155845 0.81 KMT2A (0.34) CA12
SCHEMBL7784158 0.79 ALDH1A1 (0.45) CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0894805-B1 Ribose substituted aromatic derivatives, their preparation and use as medicaments AVENTIS PHARMA SA (FR) 2005-02-09 EP disclosed
EP-0894805-A1 Ribose substituted aromatic derivatives, their preparation and use as medicaments HOECHST MARION ROUSSEL (FR) 1999-02-03 EP disclosed